Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50036057
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001435(3-Amino-N-[1-(1-{1-[2-(1-{[(1-carbamoyl-2-phenyl-e...)
Affinity DataIC50: 1nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001447(His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu-Met-NH2(Neurok...)
Affinity DataIC50: 1nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001451(CHEMBL126294 | 3-Amino-N-(1-{1-[1-({[1-(1-carbamoy...)
Affinity DataIC50: 6nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001437(CHEMBL340743 | 3-Amino-N-[1-(1-{1-[({1-[(1-carbamo...)
Affinity DataIC50: 9nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001455(CHEMBL126776 | 3-Amino-N-(1-{1-[1-(2-{1-[(1-carbam...)
Affinity DataIC50: 10nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50079412((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...)
Affinity DataIC50: 18nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001440(3-Amino-N-[1-(1-{1-[({1-[(1-carbamoyl-3-methylsulf...)
Affinity DataIC50: 50nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001454(3-Amino-N-{1-[1-(1-{[(1-{[(1-carbamoyl-3-methyl-bu...)
Affinity DataIC50: 103nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001442(CHEMBL340880 | 3-Amino-N-(1-{1-[1-(2-{1-[(1-carbam...)
Affinity DataIC50: 108nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001443(CHEMBL341015 | 3-Amino-N-[1-(1-{1-[({1-[(1-carbamo...)
Affinity DataIC50: 115nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001449(CHEMBL341065 | 3-Amino-N-(1-{1-[1-({[1-(1-carbamoy...)
Affinity DataIC50: 136nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataIC50: 148nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001444(3-Amino-N-{1-[1-(1-{[(1-{[(1-carbamoyl-3-methyl-bu...)
Affinity DataIC50: 162nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001438(3-Amino-N-{1-[1-(1-{[(1-{[(1-carbamoyl-3-methyl-bu...)
Affinity DataIC50: 193nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001453(3-Amino-N-{1-[1-(1-{[(1-{[(1-carbamoyl-3-methyl-bu...)
Affinity DataIC50: 277nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001441(CHEMBL340847 | 4-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataIC50: 1.65E+3nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001448(CHEMBL339941 | 3-Amino-N-[1-(1-{1-[({[1-(1-carbamo...)
Affinity DataIC50: 5.66E+3nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001436(CHEMBL262731 | 3-Amino-N-{1-[1-(1-{2-[1-(1-carbamo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001452(CHEMBL409334 | 3-Amino-N-(2-{1-[1-({[1-(1-carbamoy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001446(CHEMBL128175 | 3-Amino-N-(1-{1-benzyl-2-[1-({[1-(1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Golden hamster)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50001439(CHEMBL337970 | 3-Amino-N-(1-{1-[1-({[1-benzyl-2-(1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed