Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50036028
TargetMu-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001092(CHEMBL555618 | 13-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  0.900nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001092(CHEMBL555618 | 13-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  0.900nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001090(CHEMBL557749 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  2.5nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001088(CHEMBL555522 | (DPDPE)13-[2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  7nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001090(CHEMBL557749 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  9.5nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001093(CHEMBL553149 | 13-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001093(CHEMBL553149 | 13-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001093(CHEMBL553149 | 13-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  21nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001093(CHEMBL553149 | 13-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  21nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001089(CHEMBL541570 | 13-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  32nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001089(CHEMBL541570 | 13-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  32nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001089(CHEMBL541570 | 13-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  45nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001089(CHEMBL541570 | 13-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  45nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001091(CHEMBL538514 | 10-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  91nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001091(CHEMBL538514 | 10-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  91nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001091(CHEMBL538514 | 10-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  150nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001091(CHEMBL538514 | 10-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataKi:  150nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001088(CHEMBL555522 | (DPDPE)13-[2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  700nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed