Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50000058
LigandPNGBDBM50453179(CHEMBL2369463)
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000743(CHEMBL525571 | h alpha-CGRP8-37 | [Thr-His-Arg-Leu...)
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50453179(CHEMBL2369463)
Affinity DataIC50: 0.900nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000750(CHEMBL2369459 | [Val-Ala-His-Arg-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 1.70nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000750(CHEMBL2369459 | [Val-Ala-His-Arg-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 1.70nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50453179(CHEMBL2369463)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000743(CHEMBL525571 | h alpha-CGRP8-37 | [Thr-His-Arg-Leu...)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000743(CHEMBL525571 | h alpha-CGRP8-37 | [Thr-His-Arg-Leu...)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000750(CHEMBL2369459 | [Val-Ala-His-Arg-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 2.40nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000747(CHEMBL2369454 | [Arg-Leu-Ala-Gly-Leu-Leu-Ser-Arg-S...)
Affinity DataIC50: 3nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000749(CHEMBL2369458 | [Val-Thr-His-Arg-Ala-Ala-Gly-Leu-L...)
Affinity DataIC50: 8nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000749(CHEMBL2369458 | [Val-Thr-His-Arg-Ala-Ala-Gly-Leu-L...)
Affinity DataIC50: 8nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000749(CHEMBL2369458 | [Val-Thr-His-Arg-Ala-Ala-Gly-Leu-L...)
Affinity DataIC50: 8nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000742(CHEMBL2369452 | [His-Arg-Leu-Ala-Gly-Leu-Leu-Ser-A...)
Affinity DataIC50: 9nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000742(CHEMBL2369452 | [His-Arg-Leu-Ala-Gly-Leu-Leu-Ser-A...)
Affinity DataIC50: 9nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000742(CHEMBL2369452 | [His-Arg-Leu-Ala-Gly-Leu-Leu-Ser-A...)
Affinity DataIC50: 9nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000747(CHEMBL2369454 | [Arg-Leu-Ala-Gly-Leu-Leu-Ser-Arg-S...)
Affinity DataIC50: 11nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000746(CHEMBL2369457 | [Val-Thr-His-Ala-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 11nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000747(CHEMBL2369454 | [Arg-Leu-Ala-Gly-Leu-Leu-Ser-Arg-S...)
Affinity DataIC50: 12nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000746(CHEMBL2369457 | [Val-Thr-His-Ala-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 14.5nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000746(CHEMBL2369457 | [Val-Thr-His-Ala-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 15nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000744(CHEMBL2369464 | [Val-Thr-Ala-Arg-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 20nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000744(CHEMBL2369464 | [Val-Thr-Ala-Arg-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 20.2nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000744(CHEMBL2369464 | [Val-Thr-Ala-Arg-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 20.2nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000745(CHEMBL2369465 | [Val-Thr-His-Arg-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 21.9nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000745(CHEMBL2369465 | [Val-Thr-His-Arg-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 22nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50000745(CHEMBL2369465 | [Val-Thr-His-Arg-Leu-Ala-Gly-Leu-L...)
Affinity DataIC50: 25nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed