Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50037171
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130880(pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-L...)
Affinity DataIC50: 0.200nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130898(DTPA-Gly(Pip)-Pro-Arg-Gly(PipAm)-Arg-Pro-Tyr-tBuGl...)
Affinity DataIC50: 0.300nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130895(DTPA-Cha(tr-4-Mam)-Pro-Arg-Gly(PipAm)-Arg-Pro-Tyr-...)
Affinity DataIC50: 0.300nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130873(DTPA-Arg-Arg-Pro-Tur-Ile-Leu-OH | CHEMBL409477)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130899(DTPA-DLys-Pro-Arg-Gly(PipAm)-Arg-Pro-DTyr-tBuGly-L...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130876(DTPA-DTyr-Glu-Asn-Lys-Pro-Gly(PipAm)-Arg-Pro-Tyr-t...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130885(DTPA-DLys-Pro-Arg-Phe(4-Gu)-Pro-Tyr-Ile-Leu-OH | C...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130882(DTPA-DLys-Pro-Arg-Gly(PipAm)-Arg-Pro-Tyr-tBuGly-Le...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130886(alpha-FITC-Gly(Pip)-Pro-Gly(PipAm)-Arg-Pro-Tyr--tB...)
Affinity DataIC50: 0.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50370236(CHEMBL1790850)
Affinity DataIC50: 0.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130883(epsilon-FITC-DLys-Pro-Gly(PipAm)-Arg-Pro-Tyr--Ile-...)
Affinity DataIC50: 0.600nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130875(DTPA-DTyr-Glu-Asn-Lys-Pro-Gly(PipAm)-Arg-Pro-Tyr-t...)
Affinity DataIC50: 0.600nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130888(alpha-FITC-DLys-Pro-Gly(PipAm)-Arg-Pro-Tyr--Ile-Le...)
Affinity DataIC50: 1.20nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130896(DTPA-DTyr-Glu-Asn-Lys-Pro-Gly(PipAm)-Arg-Pro-Tyr-t...)
Affinity DataIC50: 1.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130878(DTPA-DLys-Pro-Arg-Ala(PipAm)-Arg-Pro-Tyr-tBuGly-Le...)
Affinity DataIC50: 2.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130893(alpha,epsilon-Bis(FITC)-DLys-Pro-Gly(PipAm)-Arg-Pr...)
Affinity DataIC50: 3.40nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130890(DTPA-DLys-Pro-Arg-hAla(PipAm)-Arg-Pro-Tyr-tBuGly-L...)
Affinity DataIC50: 6.30nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50370235(CHEMBL1790849)
Affinity DataIC50: 10.2nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130887(DTPA-DLys-ACA-Arg-Gly(PipAm)-Arg-Pro-Tyr-tBuGly-Le...)
Affinity DataIC50: 11.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130877(DTPA-DLys-Pro-Gly(PipAm)-Arg-Pro-Tyr-tBuGly-Cha-OH...)
Affinity DataIC50: 11.9nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130892(DTPA-DLys-Pro-Gly(PipAm)-Arg-Pro-Tyr-tBuGly-tBuAla...)
Affinity DataIC50: 21.7nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50370234(CHEMBL1790851)
Affinity DataIC50: 22.1nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130889(DTPA-DLys-Pro-Arg-Phe(4-Gu)-Arg-Pro-Tyr-tBuGly-Leu...)
Affinity DataIC50: 24.6nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130891(DTPA-DLys-Pro-Gly(PipAm)-Arg-Pro-Tyr-tBuGly-Cpa-OH...)
Affinity DataIC50: 42.4nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130881(DTPA-DLys-Pro-Arg-Gly(PipAm)-Gly(Pip)-Pro-Tyr-tBuG...)
Affinity DataIC50: 59.6nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130872(DTPA-DLys-Pro-Arg-Gly(PipAm)-Arg-Pro-mTyr-tBuGly-L...)
Affinity DataIC50: 106nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130897(DTPA-DLys-Pro-Arg-Gly(PipAm)-Arg-ACA-Tyr-tBuGly-Le...)
Affinity DataIC50: 113nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130879(DTPA-Ala(Pip)-Pro-Arg-Gly(PipAm)-Arg-Pro-Tyr-tBuGl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed