Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50013063
TargetMu-type opioid receptor(Guinea pig)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125999((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataIC50: 0.0340nMAssay Description:Ability to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125999((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataIC50: 0.398nMAssay Description:Ability to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126003((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50: 1.70nMAssay Description:Ability to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126000((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50: 2.80nMAssay Description:Ability to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125998((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50: 5.30nMAssay Description:Ability to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125996((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50: 9.90nMAssay Description:Ability to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125997((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50: 20nMAssay Description:Ability to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126003((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50: 28nMAssay Description:Ability to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126000((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50: 50nMAssay Description:Ability to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125998((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50: 116nMAssay Description:Ability to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125996((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50: 188nMAssay Description:Ability to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125997((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50: 305nMAssay Description:Ability to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126002((R)-2-[(R)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50: 320nMAssay Description:Ability to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126001((R)-2-((S)-2-Amino-3-phenyl-propionylamino)-5-guan...)
Affinity DataIC50: 633nMAssay Description:Ability to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126002((R)-2-[(R)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50: 1.47E+3nMAssay Description:Ability to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126001((R)-2-((S)-2-Amino-3-phenyl-propionylamino)-5-guan...)
Affinity DataIC50: 7.14E+3nMAssay Description:Ability to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125999((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  0.00205nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126000((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi:  0.0216nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126003((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  0.0350nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125997((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  0.0618nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125996((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi:  0.0623nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125998((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  0.172nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125999((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  1.10nMAssay Description:Ability to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126001((R)-2-((S)-2-Amino-3-phenyl-propionylamino)-5-guan...)
Affinity DataKi:  7.20nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126002((R)-2-[(R)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi:  7.60nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125998((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  482nMAssay Description:Ability to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126003((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  544nMAssay Description:Ability to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126000((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi:  1.69E+3nMAssay Description:Ability to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125996((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi:  2.57E+3nMAssay Description:Ability to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126002((R)-2-[(R)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi: >2.82E+3nMAssay Description:Ability to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126001((R)-2-((S)-2-Amino-3-phenyl-propionylamino)-5-guan...)
Affinity DataKi: >2.82E+3nMAssay Description:Ability to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125997((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi: >2.82E+3nMAssay Description:Ability to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed