Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50012883
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073956({5-Aminomethyl-2-[2-(9-chloro-2,3-dioxo-2,3,6,7-te...)
Affinity DataIC50: 1nMAssay Description:Affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of tritium labeled selective glycine antagonist [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123792(3-[(4-Aminomethyl-2-carboxymethyl-phenylcarbamoyl)...)
Affinity DataIC50: 1.5nMAssay Description:Affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of tritium labeled selective glycine antagonist [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123790(3-{[4-Aminomethyl-2-(1-carboxy-ethyl)-phenylcarbam...)
Affinity DataIC50: 2.70nMAssay Description:Affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of tritium labeled selective glycine antagonist [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123796(3-[(2-Carboxymethyl-phenylcarbamoyl)-methyl]-7-chl...)
Affinity DataIC50: 7.60nMAssay Description:Affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of tritium labeled selective glycine antagonist [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123791(3-[(4-Aminomethyl-phenylcarbamoyl)-methyl]-7-chlor...)
Affinity DataIC50: 18nMAssay Description:Affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of tritium labeled selective glycine antagonist [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123795(7-Chloro-3-phenylcarbamoylmethyl-1,3,4,5-tetrahydr...)
Affinity DataIC50: 19nMAssay Description:Affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of tritium labeled selective glycine antagonist [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123794(3-{[4-Aminomethyl-2-(1-carboxy-ethyl)-phenylcarbam...)
Affinity DataIC50: 29nMAssay Description:Affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of tritium labeled selective glycine antagonist [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123793(3-[(4-Aminomethyl-2-carboxymethoxy-phenylcarbamoyl...)
Affinity DataIC50: 33nMAssay Description:Affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of tritium labeled selective glycine antagonist [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123793(3-[(4-Aminomethyl-2-carboxymethoxy-phenylcarbamoyl...)
Affinity DataIC50: 33nMAssay Description:Affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of tritium labeled selective glycine antagonist [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123790(3-{[4-Aminomethyl-2-(1-carboxy-ethyl)-phenylcarbam...)
Affinity DataKi:  1nMAssay Description:Binding affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of [3H]- DCKA (5,7-dichlorokynurenic acid) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123790(3-{[4-Aminomethyl-2-(1-carboxy-ethyl)-phenylcarbam...)
Affinity DataKi:  11nMAssay Description:Binding affinity for glycine site of N-methyl-D-aspartate glutamate receptor determined by displacement of [3H]- glycine in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed