Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50012880
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataIC50: 183nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123742(Cyclosporin A analogue | CHEMBL412946)
Affinity DataIC50: 348nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assay (morn)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123747(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: 363nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123748(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: 581nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123744(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: 636nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123738(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: 742nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assay (morn)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123741(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: 840nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123743(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: 890nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123746(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: 1.54E+3nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123738(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: 1.92E+3nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assay (MOM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123742(Cyclosporin A analogue | CHEMBL412946)
Affinity DataIC50: 2.15E+3nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assay (MTM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123739(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: 5.00E+3nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123740(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: 5.00E+3nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed