Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50012610
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50116538(SC-57461A | CHEMBL543405 | CHEMBL112671 | 3-{[3-(4...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121000({2-[2-(4-Benzyl-phenoxy)-ethyl]-2-aza-bicyclo[2.2....)
Affinity DataIC50: 15nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121000({2-[2-(4-Benzyl-phenoxy)-ethyl]-2-aza-bicyclo[2.2....)
Affinity DataIC50: 15nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121003(1-[2-(4-Benzyl-phenoxy)-ethyl]-pyrrolidine-3-carbo...)
Affinity DataIC50: 16nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121009(1-[2-(4-Benzyl-phenoxy)-ethyl]-pyrrolidin-3-ylamin...)
Affinity DataIC50: 20nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50085279(1-[2-(4-Benzyl-phenoxy)-ethyl]-pyrrolidine | 1-[2-...)
Affinity DataIC50: 26nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121023(1-[2-(4-Benzyl-phenoxy)-ethyl]-pyrrolidin-3-ol | C...)
Affinity DataIC50: 30nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121010(2-[2-(4-Benzyl-phenoxy)-ethyl]-2-aza-bicyclo[2.2.1...)
Affinity DataIC50: 47nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121008(N-{1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidin-4-yl}-...)
Affinity DataIC50: 50nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121001({1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidin-4-yl}-me...)
Affinity DataIC50: 52nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50085285(1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidine | CHEMBL...)
Affinity DataIC50: 55nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121011(1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidine-4-carbox...)
Affinity DataIC50: 57nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121018({1-[2-(4-Benzyl-phenoxy)-ethyl]-pyrrolidin-3-yl}-u...)
Affinity DataIC50: 81nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121005({1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidin-4-yl}-ur...)
Affinity DataIC50: 87nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121019(({1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidine-4-carb...)
Affinity DataIC50: 110nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121007(1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidine-4-carbox...)
Affinity DataIC50: 130nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121014(N-{1-[2-(4-Benzyl-phenoxy)-ethyl]-pyrrolidin-3-yl}...)
Affinity DataIC50: 210nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121015(2-{1-[2-(4-Benzyl-phenoxy)-ethyl]-pyrrolidin-3-yl}...)
Affinity DataIC50: 210nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121017(1-[2-(4-Benzyl-phenoxy)-ethyl]-4-(1H-tetrazol-5-yl...)
Affinity DataIC50: 240nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121002(1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidine-4-carbox...)
Affinity DataIC50: 280nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121016({1-[2-(4-Benzyl-phenoxy)-ethyl]-pyrrolidin-3-yl}-a...)
Affinity DataIC50: 390nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121013((S)-1-[2-(4-Benzyl-phenoxy)-ethyl]-pyrrolidine-2-c...)
Affinity DataIC50: 450nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121004(1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidine-4-carbon...)
Affinity DataIC50: 470nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121006(4-[2-(4-Benzyl-phenoxy)-ethyl]-piperazine-1-carbox...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121020(1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidine-4-carbox...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121021(1-[2-(4-Benzyl-phenoxy)-ethyl]-piperidine-3-carbox...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50121012(1-[2-(4-Benzyl-phenoxy)-ethyl]-pyrrolidine-3-carbo...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of leukotriene A4 hydrolase in human recombinant assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed