Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50042174
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50220136(CHEMBL1471 | 5-(((2R,3S)-2-((R)-1-(3,5-bis(trifluo...)
Affinity DataIC50: 0.100nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421571(CHEMBL111303)
Affinity DataIC50: 0.794nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421552(CHEMBL108200)
Affinity DataIC50: 1nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421563(CHEMBL111176)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421562(CHEMBL108889)
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421561(CHEMBL419742)
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421564(CHEMBL107941)
Affinity DataIC50: 2.5nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421554(CHEMBL107875)
Affinity DataIC50: 3.20nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421564(CHEMBL107941)
Affinity DataIC50: 3.20nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421560(CHEMBL108667)
Affinity DataIC50: 3.20nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421573(CHEMBL321892)
Affinity DataIC50: 5nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421556(CHEMBL109183)
Affinity DataIC50: 5nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421567(CHEMBL109937)
Affinity DataIC50: 5nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM30130(Prozac | cid_62857 | Fluoxetin | CHEMBL41 | CHEMBL...)
Affinity DataIC50: 6.30nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421568(CHEMBL108422)
Affinity DataIC50: 6.30nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421558(CHEMBL432627)
Affinity DataIC50: 6.30nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421555(CHEMBL111244)
Affinity DataIC50: 7.90nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421558(CHEMBL432627)
Affinity DataIC50: 7.90nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421560(CHEMBL108667)
Affinity DataIC50: 10nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421565(CHEMBL107831)
Affinity DataIC50: 13nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421566(CHEMBL107829)
Affinity DataIC50: 13nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421553(CHEMBL320535)
Affinity DataIC50: 13nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421553(CHEMBL320535)
Affinity DataIC50: 16nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421569(CHEMBL108822)
Affinity DataIC50: 25nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421565(CHEMBL107831)
Affinity DataIC50: 25nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421563(CHEMBL111176)
Affinity DataIC50: 25nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421566(CHEMBL107829)
Affinity DataIC50: 32nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421572(CHEMBL110086)
Affinity DataIC50: 40nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421570(CHEMBL320544)
Affinity DataIC50: 50nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421570(CHEMBL320544)
Affinity DataIC50: 100nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421559(CHEMBL109514)
Affinity DataIC50: 100nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421557(CHEMBL111304)
Affinity DataIC50: 100nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421559(CHEMBL109514)
Affinity DataIC50: 158nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421562(CHEMBL108889)
Affinity DataIC50: 200nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421571(CHEMBL111303)
Affinity DataIC50: 200nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421556(CHEMBL109183)
Affinity DataIC50: 200nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421552(CHEMBL108200)
Affinity DataIC50: 200nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421573(CHEMBL321892)
Affinity DataIC50: 200nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421567(CHEMBL109937)
Affinity DataIC50: 251nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421568(CHEMBL108422)
Affinity DataIC50: 251nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421561(CHEMBL419742)
Affinity DataIC50: 251nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421572(CHEMBL110086)
Affinity DataIC50: 316nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421554(CHEMBL107875)
Affinity DataIC50: 316nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421555(CHEMBL111244)
Affinity DataIC50: 398nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421557(CHEMBL111304)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed