Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50012334
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117543(2-Amino-4-{3-methyl-1-[2-oxo-2-(toluene-4-sulfonyl...)
Affinity DataIC50: 2.00E+3nMAssay Description:Concentration required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117546(2-Amino-4-[1-(carbamoylmethyl-carbamoyl)-3-methyl-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117542(2-Amino-4-[1-(hydroxycarbamoylmethyl-carbamoyl)-3-...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibitory activity against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataIC50: 1.72E+4nMAssay Description:Concentration required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117547(2-Amino-4-[3-methyl-1-(phosphonomethyl-carbamoyl)-...)
Affinity DataIC50: 6.00E+4nMAssay Description:Concentration required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117546(2-Amino-4-[1-(carbamoylmethyl-carbamoyl)-3-methyl-...)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibitory activity against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117545(2-Amino-4-{3-methyl-1-[(1H-tetrazol-5-ylmethyl)-ca...)
Affinity DataIC50: 1.38E+5nMAssay Description:Concentration required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117542(2-Amino-4-[1-(hydroxycarbamoylmethyl-carbamoyl)-3-...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibitory constant against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117547(2-Amino-4-[3-methyl-1-(phosphonomethyl-carbamoyl)-...)
Affinity DataKi:  6.00E+4nMAssay Description:Inhibition constant was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataKi:  8.10E+4nMAssay Description:Inhibition constant was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataKi:  8.10E+4nMAssay Description:Inhibition constant was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed