Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50012324
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117496(H-His-Ala-Lys-Arg-Arg-Leu-Ile-(L)-Pse-OH | CHEMBL4...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117492(H-His-Ala-Lys-Arg-Arg-Leu-Ile-(L)-Phe omegaCH2OH |...)
Affinity DataIC50: 24nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117488(H-His-Ala-Lys-Arg-Arg-Leu-Ile-Phe-NH2 | CHEMBL2173...)
Affinity DataIC50: 39nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117490(H-His-Ala-Lys-Arg-Arg-Leu-Ile-(Z)-Dhp-OH | CHEMBL3...)
Affinity DataIC50: 70nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117487(H-His-Ala-Lys-Arg-Arg-Leu-Ile-(D)-Pse-(Ac)-OH | CH...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117499(H-His-Ala-Lys-Arg-Arg-Leu-Ile-(D)-Pse-OH | CHEMBL4...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117495(H-His-Ala-Lys-Arg-Arg-Leu-Ile-(L)-Pse-(Ac)-OH | CH...)
Affinity DataIC50: 320nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117494(H-His-Ser-Lys-Arg-Arg-Leu-Ile-(L)-Phe omegaCH2OH |...)
Affinity DataIC50: 430nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117497(H-His-Ser-Lys-Arg-Arg-Leu-Ile-(L)-Pse-OH | CHEMBL2...)
Affinity DataIC50: 560nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117498(H-His-Ser-Lys-Arg-Arg-Leu-Ile-(D)-Pse-OH | CHEMBL4...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117491(H-His-Ser-Lys-Arg-Arg-Leu-Ile-(Z)-Dhp-OH | CHEMBL2...)
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117493(H-His-Ser-Lys-Arg-Arg-Leu-Ile-Phe-NH2 | CHEMBL2369...)
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed