Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50035240
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine (-) | methyl (1R,2R,3S,5S)-3-(benzoyloxy)-...)
Affinity DataKi:  130nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine (-) | methyl (1R,2R,3S,5S)-3-(benzoyloxy)-...)
Affinity DataKi:  460nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116317(Benzhydryl-(2-phenyl-quinazolin-4-yl)-amine | CHEM...)
Affinity DataKi:  530nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116318(CHEMBL72703 | cid_5051334 | (1-Phenyl-ethyl)-(2-ph...)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116316(4-(8-Methyl-8-aza-bicyclo[3.2.1]oct-3-yloxy)-2-phe...)
Affinity DataKi:  5.10E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116316(4-(8-Methyl-8-aza-bicyclo[3.2.1]oct-3-yloxy)-2-phe...)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116319((2,2-Diphenyl-ethyl)-(2-phenyl-quinazolin-4-yl)-am...)
Affinity DataKi:  5.40E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116315(Dimethyl-[3-(2-phenyl-quinazolin-4-ylsulfanyl)-pro...)
Affinity DataKi:  6.10E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116320((1-Phenyl-ethyl)-(2-phenyl-quinazolin-4-yl)-amine ...)
Affinity DataKi:  6.10E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50033296(Benzyl-(2-phenyl-quinazolin-4-yl)-amine | CHEMBL72...)
Affinity DataKi:  7.90E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116314(4-(1-Methyl-piperidin-4-yloxy)-2-phenyl-quinazolin...)
Affinity DataKi:  9.10E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116315(Dimethyl-[3-(2-phenyl-quinazolin-4-ylsulfanyl)-pro...)
Affinity DataKi:  9.60E+3nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116324(Dimethyl-[3-(2-phenyl-quinazolin-4-yloxy)-propyl]-...)
Affinity DataKi:  9.90E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116322(N,N-Dimethyl-N'-(2-phenyl-quinazolin-4-yl)-propane...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116319((2,2-Diphenyl-ethyl)-(2-phenyl-quinazolin-4-yl)-am...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116314(4-(1-Methyl-piperidin-4-yloxy)-2-phenyl-quinazolin...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116323(4-Benzhydrylsulfanyl-2-phenyl-quinazoline | CHEMBL...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116321((3,3-Diphenyl-propyl)-(2-phenyl-quinazolin-4-yl)-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50033296(Benzyl-(2-phenyl-quinazolin-4-yl)-amine | CHEMBL72...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116322(N,N-Dimethyl-N'-(2-phenyl-quinazolin-4-yl)-propane...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116324(Dimethyl-[3-(2-phenyl-quinazolin-4-yloxy)-propyl]-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116323(4-Benzhydrylsulfanyl-2-phenyl-quinazoline | CHEMBL...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116320((1-Phenyl-ethyl)-(2-phenyl-quinazolin-4-yl)-amine ...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116321((3,3-Diphenyl-propyl)-(2-phenyl-quinazolin-4-yl)-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116317(Benzhydryl-(2-phenyl-quinazolin-4-yl)-amine | CHEM...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50116318(CHEMBL72703 | cid_5051334 | (1-Phenyl-ethyl)-(2-ph...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]RTI-55 binding to Serotonin transporter of rat caudate membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed