Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50037029
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095151((S)-2-[(S)-2-(2-{1-[(S)-2-Amino-3-((S)-4-hydroxy-p...)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataIC50: 9.90nMAssay Description:Inhibitory activity against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114009(1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrroli...)
Affinity DataIC50: 23.3nMAssay Description:Inhibitory activity against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095154((S)-2-[(S)-2-(2-{1-[(R)-2-Amino-3-((S)-4-hydroxy-p...)
Affinity DataIC50: 79nMAssay Description:Inhibitory activity against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114010(1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrroli...)
Affinity DataIC50: 80.1nMAssay Description:Inhibitory activity against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity towards Opioid receptor mu 1 by displacing [3H]DAMGO in rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards Opioid receptor mu 1 by displacing [3H]DAMGO in rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095151((S)-2-[(S)-2-(2-{1-[(S)-2-Amino-3-((S)-4-hydroxy-p...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity towards Opioid receptor mu 1 by displacing [3H]DAMGO in rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095154((S)-2-[(S)-2-(2-{1-[(R)-2-Amino-3-((S)-4-hydroxy-p...)
Affinity DataKi:  67nMAssay Description:Binding affinity towards Opioid receptor mu 1 by displacing [3H]DAMGO in rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114009(1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrroli...)
Affinity DataKi:  73nMAssay Description:Binding affinity towards Opioid receptor mu 1 by displacing [3H]DAMGO in rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114010(1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrroli...)
Affinity DataKi:  79nMAssay Description:Binding affinity towards Opioid receptor mu 1 by displacing [3H]DAMGO in rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed