Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50011746
TargetGlucagon receptor(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110054(3-Cyano-4-hydroxy-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity against rat glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110054(3-Cyano-4-hydroxy-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110068(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50: 23nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110056(2,3-Dichloro-4-hydroxy-benzoic acid [1-[4-(4-isopr...)
Affinity DataIC50: 31nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110067(2,3-Difluoro-4-hydroxy-benzoic acid [1-[4-(4-isopr...)
Affinity DataIC50: 48nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110073(4-Hydroxy-3-nitro-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50: 50nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110074(3-Chloro-4-hydroxy-benzoic acid [4-(4-isopropyl-be...)
Affinity DataIC50: 53nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110066(3-Chloro-4-hydroxy-benzoic acid [4-(4-trifluoromet...)
Affinity DataIC50: 58nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110055(3-Chloro-4-hydroxy-benzoic acid [1-(4-isopropyl-be...)
Affinity DataIC50: 84nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110057(3-Fluoro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110084(2-{4-[(3-Chloro-4-hydroxy-benzoyl)-hydrazonomethyl...)
Affinity DataIC50: 130nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110070(3-Chloro-4-hydroxy-benzoic acid [1-[4-(tetrahydro-...)
Affinity DataIC50: 140nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110063(3-Chloro-4-hydroxy-benzoic acid [1-[4-(3,4-difluor...)
Affinity DataIC50: 150nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110053(3-Chloro-4-hydroxy-benzoic acid [1-[4-(5-tert-buty...)
Affinity DataIC50: 160nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110080(3-Chloro-4-hydroxy-benzoic acid [1-[3,5-dimethoxy-...)
Affinity DataIC50: 180nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50104096(3-Chloro-4-hydroxy-benzoic acid (4-hydroxy-naphtha...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110077(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50: 330nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110083(3-Chloro-4-hydroxy-benzoic acid [1-[1-(4-isopropyl...)
Affinity DataIC50: 390nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110081({4-[(3-Chloro-4-hydroxy-benzoyl)-hydrazonomethyl]-...)
Affinity DataIC50: 690nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110071(N'-(4-(4-isopropylbenzyloxy)-3,5-dimethoxybenzylid...)
Affinity DataIC50: 690nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110085(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50: 740nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110062(3-Chloro-4-hydroxy-benzoic acid [1-(4-methoxy-naph...)
Affinity DataIC50: 870nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110060(N'-(4-(4-isopropylbenzyloxy)-3,5-dimethoxybenzyl)-...)
Affinity DataIC50: 880nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110076(3-Amino-4-hydroxy-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50: 940nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110065(2-{4-[(3-Chloro-4-hydroxy-benzoyl)-hydrazonomethyl...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110082(N'-(4-(4-isopropylbenzyloxy)-3-methoxybenzylidene)...)
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110078(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110069(3-Chloro-4-hydroxy-N-{2-[4-(4-isopropyl-benzyloxy)...)
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110058(3,4-Dihydroxy-benzoic acid [1-[4-(4-isopropyl-benz...)
Affinity DataIC50: 2.70E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110059(3-Chloro-4-hydroxy-N-{2-[4-(4-isopropyl-benzyloxy)...)
Affinity DataIC50: 5.20E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110072((E)-N-(3-Chloro-4-hydroxy-phenyl)-3-[4-(4-isopropy...)
Affinity DataIC50: 6.40E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110079(3-Cyano-4-hydroxy-benzoic acid (4-isopropyl-3,5-di...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110064(5-[(3-Chloro-4-hydroxy-benzoyl)-hydrazonomethyl]-2...)
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110061(2-chloro-4-[1-[4-(4-isopropylbenzyloxy)-3,5-dimeth...)
Affinity DataIC50: 7.83E+4nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110075(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed