Compile Data Set for Download or QSAR
Report error Found 113 Enz. Inhib. hit(s) with all data for entry = 50041052
TargetD(3) dopamine receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403975(CHEMBL315772)
Affinity DataIC50: 0.550nMAssay Description:Binding affinity for human cloned Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403975(CHEMBL315772)
Affinity DataIC50: 1nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403974(CHEMBL84931)
Affinity DataIC50: 1.10nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403974(CHEMBL84931)
Affinity DataIC50: 1.10nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403992(CHEMBL84081)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403991(CHEMBL315834)
Affinity DataIC50: 1.70nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403975(CHEMBL315772)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403986(CHEMBL82966)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(4) dopamine receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403975(CHEMBL315772)
Affinity DataIC50: 2.60nMAssay Description:Binding affinity for human cloned Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403974(CHEMBL84931)
Affinity DataIC50: 2.60nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403978(CHEMBL85735)
Affinity DataIC50: 3nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403978(CHEMBL85735)
Affinity DataIC50: 3.10nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403975(CHEMBL315772)
Affinity DataIC50: 3.5nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403983(CHEMBL314885)
Affinity DataIC50: 3.80nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403984(CHEMBL82635)
Affinity DataIC50: 3.90nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403992(CHEMBL84081)
Affinity DataIC50: 4.70nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403991(CHEMBL315834)
Affinity DataIC50: 5nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403978(CHEMBL85735)
Affinity DataIC50: 5.90nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403984(CHEMBL82635)
Affinity DataIC50: 6nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403976(CHEMBL314107)
Affinity DataIC50: 6.20nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403977(CHEMBL85155)
Affinity DataIC50: 6.30nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146360(Dimethyl-[(2S,3aR)-1-(2,3,3a,8-tetrahydro-1-oxa-12...)
Affinity DataIC50: 6.80nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403992(CHEMBL84081)
Affinity DataIC50: 6.90nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403981(CHEMBL84810)
Affinity DataIC50: 7.60nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403987(CHEMBL315308)
Affinity DataIC50: 7.90nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403975(CHEMBL315772)
Affinity DataIC50: 8.70nMAssay Description:Binding affinity for human cloned Dopamine receptor D2LMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Rat)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403975(CHEMBL315772)
Affinity DataIC50: 8.90nMAssay Description:Binding affinity for rat Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403977(CHEMBL85155)
Affinity DataIC50: 10nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403979(CHEMBL313604)
Affinity DataIC50: 10nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403983(CHEMBL314885)
Affinity DataIC50: 11nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403976(CHEMBL314107)
Affinity DataIC50: 11nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403987(CHEMBL315308)
Affinity DataIC50: 11nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146360(Dimethyl-[(2S,3aR)-1-(2,3,3a,8-tetrahydro-1-oxa-12...)
Affinity DataIC50: 12nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403986(CHEMBL82966)
Affinity DataIC50: 12nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403990(CHEMBL314795)
Affinity DataIC50: 12nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403974(CHEMBL84931)
Affinity DataIC50: 14nMAssay Description:Binding affinity for human cloned Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(4) dopamine receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403974(CHEMBL84931)
Affinity DataIC50: 14nMAssay Description:Binding affinity for human cloned Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403975(CHEMBL315772)
Affinity DataIC50: 14nMAssay Description:Binding affinity for human cloned Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403980(CHEMBL315044)
Affinity DataIC50: 14nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403979(CHEMBL313604)
Affinity DataIC50: 15nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403977(CHEMBL85155)
Affinity DataIC50: 16nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403976(CHEMBL314107)
Affinity DataIC50: 17nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403980(CHEMBL315044)
Affinity DataIC50: 19nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM31005(MIANSERIN HYDROCHLORIDE | SMR000058472 | MLS000069...)
Affinity DataIC50: 21nMAssay Description:Binding affinity for human cloned Alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403987(CHEMBL315308)
Affinity DataIC50: 22nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146360(Dimethyl-[(2S,3aR)-1-(2,3,3a,8-tetrahydro-1-oxa-12...)
Affinity DataIC50: 23nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403991(CHEMBL315834)
Affinity DataIC50: 24nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403990(CHEMBL314795)
Affinity DataIC50: 30nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403986(CHEMBL82966)
Affinity DataIC50: 32nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50403979(CHEMBL313604)
Affinity DataIC50: 32nMAssay Description:Binding affinity for human cloned 5-HT2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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