Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50011057
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101787(4-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101782(4-Nitro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEM...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(LUF-5417 | 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101783(4-Bromo-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEM...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101781(4-Methyl-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101790(N-(4-Phenyl-thiazol-2-yl)-benzamide | CHEMBL60334)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101786(2,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide |...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101784(3,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide |...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097446(4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide ...)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(LUF-5417 | 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101789(3-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101788(N-(4-Phenyl-thiazol-2-yl)-4-trifluoromethyl-benzam...)
Affinity DataKi:  165nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  670nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101785(4-tert-Butyl-N-(4-phenyl-thiazol-2-yl)-benzamide |...)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]ZM-241385 from A2A receptor in rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097446(4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide ...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed