Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50011022
LigandPNGBDBM50101427((R)-2-(5-nitro-1H-indol-3-yl)-2-oxo-N-(1-phenyleth...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-1-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50101429(2-(1H-Indol-3-yl)-N-(4-nitro-benzyl)-2-oxo-acetami...)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-1-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50066949((1H-Indol-3-yl)-oxo-acetic acid N'-(4-nitro-phenyl...)
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-1-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50066949((1H-Indol-3-yl)-oxo-acetic acid N'-(4-nitro-phenyl...)
Affinity DataKi:  40nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-3-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50055247(N-(4-methoxybenzyl)-2-(5-nitro-1H-indol-3-yl)-2-ox...)
Affinity DataKi:  42nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-1-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50066949((1H-Indol-3-yl)-oxo-acetic acid N'-(4-nitro-phenyl...)
Affinity DataKi:  43nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-5-beta-3-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM26266(Ambien | CHEMBL911 | ZPM | N,N-dimethyl-2-[6-methy...)
Affinity DataKi:  50nMAssay Description:Inhibition of [3H]flumazenil specific binding at rat GABA-A alpha-1-beta-2-gamma-2 receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50101429(2-(1H-Indol-3-yl)-N-(4-nitro-benzyl)-2-oxo-acetami...)
Affinity DataKi:  58nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-5-beta-3-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50268784((R)-N-(2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-in...)
Affinity DataKi:  95nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-5-beta-3-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50055247(N-(4-methoxybenzyl)-2-(5-nitro-1H-indol-3-yl)-2-ox...)
Affinity DataKi:  126nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-5-beta-3-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50055247(N-(4-methoxybenzyl)-2-(5-nitro-1H-indol-3-yl)-2-ox...)
Affinity DataKi:  137nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-3-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50089770(1-(1,3-Dihydro-isoindol-2-yl)-2-(1H-indol-3-yl)-et...)
Affinity DataKi:  224nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-1-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50101427((R)-2-(5-nitro-1H-indol-3-yl)-2-oxo-N-(1-phenyleth...)
Affinity DataKi:  239nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-5-beta-3-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50101427((R)-2-(5-nitro-1H-indol-3-yl)-2-oxo-N-(1-phenyleth...)
Affinity DataKi:  283nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-3-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM26266(Ambien | CHEMBL911 | ZPM | N,N-dimethyl-2-[6-methy...)
Affinity DataKi:  765nMAssay Description:Inhibition of [3H]-flumazenil binding to rat GABA-A receptor alpha-3-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50101422(2-(1H-Indol-3-yl)-2-oxo-N-(1-phenyl-ethyl)-acetami...)
Affinity DataKi:  1.15E+3nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-1-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50101429(2-(1H-Indol-3-yl)-N-(4-nitro-benzyl)-2-oxo-acetami...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-3-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50268784((R)-N-(2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-in...)
Affinity DataKi:  1.96E+3nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-3-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50268744((R)-N-(2,3-dihydro-1H-inden-1-yl)-2-(1H-indol-3-yl...)
Affinity DataKi:  2.16E+3nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-5-beta-3-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50089770(1-(1,3-Dihydro-isoindol-2-yl)-2-(1H-indol-3-yl)-et...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-3-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50101422(2-(1H-Indol-3-yl)-2-oxo-N-(1-phenyl-ethyl)-acetami...)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition of [3H]flumazenil binding to rat alpha-5-beta-3-gamma-2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed