Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 5316
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50019492(RX821002 | CHEMBL10332 | 2-(2-methoxy-2,3-dihydrob...)
Affinity DataKi:  0.920nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50019492(RX821002 | CHEMBL10332 | 2-(2-methoxy-2,3-dihydrob...)
Affinity DataKi:  0.950nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  3.70nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  4.5nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  4.90nMMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  5.30nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50019492(RX821002 | CHEMBL10332 | 2-(2-methoxy-2,3-dihydrob...)
Affinity DataKi:  6.40nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50019492(RX821002 | CHEMBL10332 | 2-(2-methoxy-2,3-dihydrob...)
Affinity DataKi:  7.30nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  11.3nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  11.8nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  13.5nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM81773(BAM-1303 | CAS_115219-10-8 | BAM 1303)
Affinity DataKi:  18.1nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  18.4nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  21.5nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  24.1nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  28.3nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50030623(SK&F-104078 | SK-104078 | SKF 104078 | CHEMBL11416...)
Affinity DataKi:  30.4nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  37nMMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM81773(BAM-1303 | CAS_115219-10-8 | BAM 1303)
Affinity DataKi:  46nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM30993(Ajmalicine | MLS000111555 | SMR000107477 | Raubasi...)
Affinity DataKi:  47.6nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataKi:  57nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  63.6nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  66nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  92nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM81773(BAM-1303 | CAS_115219-10-8 | BAM 1303)
Affinity DataKi:  95.3nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  129nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  142nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  169nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50030623(SK&F-104078 | SK-104078 | SKF 104078 | CHEMBL11416...)
Affinity DataKi:  191nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50030623(SK&F-104078 | SK-104078 | SKF 104078 | CHEMBL11416...)
Affinity DataKi:  244nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataKi:  284nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50030623(SK&F-104078 | SK-104078 | SKF 104078 | CHEMBL11416...)
Affinity DataKi:  292nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM81773(BAM-1303 | CAS_115219-10-8 | BAM 1303)
Affinity DataKi:  313nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM81772(NSC_122211 | CAS_122211 | ARC-239)
Affinity DataKi:  373nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM30993(Ajmalicine | MLS000111555 | SMR000107477 | Raubasi...)
Affinity DataKi:  376nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Rabbit)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM30993(Ajmalicine | MLS000111555 | SMR000107477 | Raubasi...)
Affinity DataKi:  429nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM81772(NSC_122211 | CAS_122211 | ARC-239)
Affinity DataKi:  484nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataKi:  558nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  722nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataKi:  913nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataKi:  996nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataKi:  1.03E+3nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM30993(Ajmalicine | MLS000111555 | SMR000107477 | Raubasi...)
Affinity DataKi:  1.47E+3nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  2.13E+3nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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