Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50010794
TargetPotassium voltage-gated channel subfamily A member 3(Mouse)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50083523([1-Benzyl-1H-quinolin-(4E)-ylidene]-pentyl-amine |...)
Affinity DataIC50: 230nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Mouse)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50098785(4-Benzhydryloxymethyl-1-[3-(4-methoxy-phenyl)-prop...)
Affinity DataIC50: 280nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Mouse)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50098782(2-Isopropyl-8-methoxy-5-methyl-5H-furo[3,2-c]quino...)
Affinity DataIC50: 5.00E+3nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Mouse)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50098781(9-Methoxy-2,2,6-trimethyl-2,6-dihydro-pyrano[3,2-c...)
Affinity DataIC50: 1.00E+4nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Mouse)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50098784(9-Methoxy-2,2,6-trimethyl-2,3,4,6-tetrahydro-pyran...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of voltage-gated potassium channel subunit Kv1.3 expressed in L929 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Mouse)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50098783(kokusaginine | 4,6,7-Trimethoxy-furo[2,3-b]quinoli...)
Affinity DataIC50: 4.90E+4nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed