Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50023368
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50241525(3-O-acetyl-9,11-dehydro-beta-boswellic acid | CHEM...)
Affinity DataIC50: 750nMAssay Description:Inhibition of lipoxygenase 5 product formation from endogenous substrate in Calcium and ionophore-stimulated polymorphonuclear leukocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50241262(3-O-acetyl-11-keto-beta-boswellic acid | 3alpha-ac...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of lipoxygenase 5 product formation from endogenous substrate in Calcium and ionophore-stimulated polymorphonuclear leukocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50241261(11-keto-beta-boswellicacid | (3R,4R,4aR,6aR,6bS,8a...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of lipoxygenase 5 product formation from endogenous substrate in Calcium and ionophore-stimulated polymorphonuclear leukocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed