Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50036818
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089269(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[3-(1H-indol-3...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061828(N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[3-(1H-indol-...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089268(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-(4...)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0900nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089276(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[3-(1H-indol-3...)
Affinity DataKi:  0.980nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089275(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-(4...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089277(N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[2-(2-{2-[2-(...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089272(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[3-(1H-indol-3...)
Affinity DataKi:  19nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089275(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-(4...)
Affinity DataKi:  36nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089270(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-(4...)
Affinity DataKi:  51nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089276(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[3-(1H-indol-3...)
Affinity DataKi:  84nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089269(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[3-(1H-indol-3...)
Affinity DataKi:  123nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089272(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[3-(1H-indol-3...)
Affinity DataKi:  150nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089268(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-(4...)
Affinity DataKi:  200nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061828(N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[3-(1H-indol-...)
Affinity DataKi:  224nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089277(N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[2-(2-{2-[2-(...)
Affinity DataKi:  960nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed