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Found
26
Enz. Inhib. hit(s) with all data for entry = 5263
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM21397
(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
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Affinity Data
Ki: 0.275nM
More data for this Ligand-Target Pair
Target Info
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ChEBI
CHEMBL
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PC sid
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Article
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PubMed
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Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM21397
(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.295nM
More data for this Ligand-Target Pair
Target Info
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UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
PC cid
PC sid
PDB
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In Depth
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Article
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PubMed
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Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM85672
(S33084)
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Affinity Data
Ki: 0.302nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM85672
(S33084)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.372nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM21397
(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.710nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM85672
(S33084)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.933nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50240797
(GR218231 | [6-(4-Methoxy-benzenesulfonylmethyl)-1,...)
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Affinity Data
Ki: 1.12nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50240797
(GR218231 | [6-(4-Methoxy-benzenesulfonylmethyl)-1,...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.38nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50240797
(GR218231 | [6-(4-Methoxy-benzenesulfonylmethyl)-1,...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.95nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50010586
(CHEMBL70565 | (-)-1-Propyl-2,3,10,10a-tetrahydro-1...)
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Affinity Data
Ki: 2.14nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
PDB
3D Structure (crystal)
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50020222
(CHEMBL285755 | 7-Dipropylamino-5,6,7,8-tetrahydro-...)
Copy SMILES
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Affinity Data
Ki: 2.19nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM21398
(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Copy SMILES
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Affinity Data
Ki: 2.19nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
DrugBank
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50010586
(CHEMBL70565 | (-)-1-Propyl-2,3,10,10a-tetrahydro-1...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.55nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
PDB
3D Structure (crystal)
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM21398
(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.98nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
DrugBank
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50020222
(CHEMBL285755 | 7-Dipropylamino-5,6,7,8-tetrahydro-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4.37nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50010586
(CHEMBL70565 | (-)-1-Propyl-2,3,10,10a-tetrahydro-1...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 7.59nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
PDB
3D Structure (crystal)
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM21398
(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 10nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
DrugBank
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50133937
(CHEMBL140184 | S14297 | (2,3,5,6,7,8-Hexahydro-nap...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 11.5nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50133937
(CHEMBL140184 | S14297 | (2,3,5,6,7,8-Hexahydro-nap...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 12.3nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM50133937
(CHEMBL140184 | S14297 | (2,3,5,6,7,8-Hexahydro-nap...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 33.1nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM55121
(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 33.9nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
DrugBank
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM55121
(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 55.0nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
DrugBank
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM55121
(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 104nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
DrugBank
KEGG
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM22869
(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 245nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM22869
(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 562nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
D(3) dopamine receptor
(Human)
Croissy-Sur-Seine Paris
Curated by
PDSP K
i
Database
Ligand
BDBM22869
(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 708nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
ChEBI
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
PubMed
Copy reaction URL