Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50036901
TargetSubstance-P receptor(Human)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369778(CHEMBL1791164)
Affinity DataIC50: 165nMAssay Description:Compound was tested for delta antagonist activity against tachykinin NK-1.Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369779(CHEMBL1791163)
Affinity DataIC50: 216nMAssay Description:Compound was tested for delta antagonist activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369780(CHEMBL1791161)
Affinity DataIC50: 1.05E+3nMAssay Description:Compound was tested for delta antagonist activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50085050(H-Dmt-c [-D-Orn-2-Nal-D-Pro-Gly-] | CHEMBL152690)
Affinity DataKi:  0.467nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50085050(H-Dmt-c [-D-Orn-2-Nal-D-Pro-Gly-] | CHEMBL152690)
Affinity DataKi:  0.476nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50085049(CHO-Dmt-c [-D-Orn-2-Nal-D-Pro-Gly-] | CHEMBL152689)
Affinity DataKi:  32.8nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50085055(Dhp-c-[-D-Orn-2-Nal-D-Pro-Gly-] | CHEMBL151098)
Affinity DataKi:  109nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369778(CHEMBL1791164)
Affinity DataKi:  152nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50085049(CHO-Dmt-c [-D-Orn-2-Nal-D-Pro-Gly-] | CHEMBL152689)
Affinity DataKi:  218nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50085055(Dhp-c-[-D-Orn-2-Nal-D-Pro-Gly-] | CHEMBL151098)
Affinity DataKi:  450nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369779(CHEMBL1791163)
Affinity DataKi:  486nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369780(CHEMBL1791161)
Affinity DataKi:  759nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369777(CHEMBL1791165)
Affinity DataKi:  1.07E+3nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369779(CHEMBL1791163)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369780(CHEMBL1791161)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369778(CHEMBL1791164)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montr£Al

Curated by ChEMBL
LigandPNGBDBM50369777(CHEMBL1791165)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed