Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50009539
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084952(4'-Carbamimidoyl-2'-methyl-biphenyl-4-carboxylic a...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084958(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 0.930nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084953(2-Methyl-biphenyl-4,4'-dicarboxylic acid 4-amide 4...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM79215(SMR001230745 | N-[4-methoxy-3-(4-methylpiperazin-1...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084959(4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)pheny...)
Affinity DataIC50: 2nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084952(4'-Carbamimidoyl-2'-methyl-biphenyl-4-carboxylic a...)
Affinity DataIC50: 3nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084961(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 6.30nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084960(2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biph...)
Affinity DataIC50: 7.30nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084953(2-Methyl-biphenyl-4,4'-dicarboxylic acid 4-amide 4...)
Affinity DataIC50: 10nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084951(2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biph...)
Affinity DataIC50: 10nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084952(4'-Carbamimidoyl-2'-methyl-biphenyl-4-carboxylic a...)
Affinity DataIC50: 23nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084958(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 37nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM79215(SMR001230745 | N-[4-methoxy-3-(4-methylpiperazin-1...)
Affinity DataIC50: 52nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084953(2-Methyl-biphenyl-4,4'-dicarboxylic acid 4-amide 4...)
Affinity DataIC50: 57nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084955(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 60nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084954(Methanesulfonic acid 4-{[2'-methyl-4'-(5-methyl-[1...)
Affinity DataIC50: 70nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084961(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 100nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084961(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 400nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084952(4'-Carbamimidoyl-2'-methyl-biphenyl-4-carboxylic a...)
Affinity DataIC50: 407nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM79215(SMR001230745 | N-[4-methoxy-3-(4-methylpiperazin-1...)
Affinity DataIC50: 425nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084960(2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biph...)
Affinity DataIC50: 467nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084951(2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biph...)
Affinity DataIC50: 600nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084957(Trifluoro-methanesulfonic acid 4-{[2'-methyl-4'-(5...)
Affinity DataIC50: 700nMAssay Description:Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084955(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 700nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084955(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 700nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084951(2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biph...)
Affinity DataIC50: 900nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084959(4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)pheny...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084957(Trifluoro-methanesulfonic acid 4-{[2'-methyl-4'-(5...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084954(Methanesulfonic acid 4-{[2'-methyl-4'-(5-methyl-[1...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084955(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084960(2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM79215(SMR001230745 | N-[4-methoxy-3-(4-methylpiperazin-1...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084960(2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084958(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084953(2-Methyl-biphenyl-4,4'-dicarboxylic acid 4-amide 4...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084957(Trifluoro-methanesulfonic acid 4-{[2'-methyl-4'-(5...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084958(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084959(4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)pheny...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084954(Methanesulfonic acid 4-{[2'-methyl-4'-(5-methyl-[1...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084961(2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biph...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084959(4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)pheny...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084951(2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biph...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084954(Methanesulfonic acid 4-{[2'-methyl-4'-(5-methyl-[1...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50084957(Trifluoro-methanesulfonic acid 4-{[2'-methyl-4'-(5...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assaysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed