Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50036900
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50064106({[(S)-2-Biphenyl-4-yl-1-(2H-tetrazol-5-yl)-ethylam...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084905({1-[2-Dibenzofuran-3-yl-1-(1H-tetrazol-5-yl)-ethyl...)
Affinity DataIC50: 2.60nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084905({1-[2-Dibenzofuran-3-yl-1-(1H-tetrazol-5-yl)-ethyl...)
Affinity DataIC50: 2.60nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084897(3-Dibenzofuran-3-yl-2-[3-dibenzofuran-3-yl-2-(phos...)
Affinity DataIC50: 2.70nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM21641(2-(2-benzyl-3-sulfanylpropanamido)acetic acid | CH...)
Affinity DataIC50: 4.80nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50064109({1-[2-Biphenyl-4-yl-1-(1H-tetrazol-5-yl)-ethylamin...)
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084903({[2-Dibenzofuran-3-yl-1-(1H-tetrazol-5-yl)-ethylam...)
Affinity DataIC50: 6nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084897(3-Dibenzofuran-3-yl-2-[3-dibenzofuran-3-yl-2-(phos...)
Affinity DataIC50: 6.40nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50064110(CHEMBL147847 | 2-{2-[(S)-5-(2,4-Difluoro-phenyl)-2...)
Affinity DataIC50: 8nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084895(2-[3-Dibenzofuran-3-yl-2-(phosphonomethyl-amino)-p...)
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084898(2-[3-Dibenzofuran-3-yl-2-(phosphonomethyl-amino)-p...)
Affinity DataIC50: 13nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50064096({[(S)-4-(2-Fluoro-phenyl)-1-(2H-tetrazol-5-yl)-but...)
Affinity DataIC50: 14nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50064109({1-[2-Biphenyl-4-yl-1-(1H-tetrazol-5-yl)-ethylamin...)
Affinity DataIC50: 17nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084893(3-Dibenzofuran-3-yl-2-(phosphonomethyl-amino)-prop...)
Affinity DataIC50: 22nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084892(3-Dibenzofuran-3-yl-2-[1-phosphono-3-(3,4,5-trimet...)
Affinity DataIC50: 22nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084895(2-[3-Dibenzofuran-3-yl-2-(phosphonomethyl-amino)-p...)
Affinity DataIC50: 23nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084910(3-Dibenzofuran-3-yl-2-[3-(3,4-dimethoxy-phenyl)-1-...)
Affinity DataIC50: 29nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084910(3-Dibenzofuran-3-yl-2-[3-(3,4-dimethoxy-phenyl)-1-...)
Affinity DataIC50: 29nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50251742((S)-2-{(R)-2-[Hydroxy-((2R,3R,4R,5R,6S)-3,4,5-trih...)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084911({[2-(9-Oxo-9H-fluoren-2-yl)-1-(1H-tetrazol-5-yl)-e...)
Affinity DataIC50: 30nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084898(2-[3-Dibenzofuran-3-yl-2-(phosphonomethyl-amino)-p...)
Affinity DataIC50: 31nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084912(3-Dibenzofuran-3-yl-2-[1-phosphono-3-(2,4,5-trimet...)
Affinity DataIC50: 40nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50064120((S)-2-[(S)-5-(2,4-Difluoro-phenyl)-2-(phosphonomet...)
Affinity DataIC50: 51nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084900(3-Dibenzofuran-3-yl-2-(5-methyl-1-phosphono-hexyla...)
Affinity DataIC50: 65nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084899(2-(5-Amino-1-phosphono-pentylamino)-3-dibenzofuran...)
Affinity DataIC50: 97nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084894(3-Dibenzofuran-3-yl-2-[3-(2,3-dimethoxy-phenyl)-1-...)
Affinity DataIC50: 110nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084894(3-Dibenzofuran-3-yl-2-[3-(2,3-dimethoxy-phenyl)-1-...)
Affinity DataIC50: 110nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084903({[2-Dibenzofuran-3-yl-1-(1H-tetrazol-5-yl)-ethylam...)
Affinity DataIC50: 114nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084909({[2-(9-Methyl-9H-carbazol-2-yl)-1-(1H-tetrazol-5-y...)
Affinity DataIC50: 140nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50064096({[(S)-4-(2-Fluoro-phenyl)-1-(2H-tetrazol-5-yl)-but...)
Affinity DataIC50: 150nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084896(3-Dibenzofuran-3-yl-2-(1-phosphono-ethylamino)-pro...)
Affinity DataIC50: 180nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084896(3-Dibenzofuran-3-yl-2-(1-phosphono-ethylamino)-pro...)
Affinity DataIC50: 180nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084891(3-Dibenzofuran-3-yl-2-(1-phosphono-3-quinolin-8-yl...)
Affinity DataIC50: 200nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084891(3-Dibenzofuran-3-yl-2-(1-phosphono-3-quinolin-8-yl...)
Affinity DataIC50: 200nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084905({1-[2-Dibenzofuran-3-yl-1-(1H-tetrazol-5-yl)-ethyl...)
Affinity DataIC50: 210nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084905({1-[2-Dibenzofuran-3-yl-1-(1H-tetrazol-5-yl)-ethyl...)
Affinity DataIC50: 210nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084911({[2-(9-Oxo-9H-fluoren-2-yl)-1-(1H-tetrazol-5-yl)-e...)
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50064106({[(S)-2-Biphenyl-4-yl-1-(2H-tetrazol-5-yl)-ethylam...)
Affinity DataIC50: 410nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084906({[2-(9H-Fluoren-2-yl)-1-(1H-tetrazol-5-yl)-ethylam...)
Affinity DataIC50: 450nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084906({[2-(9H-Fluoren-2-yl)-1-(1H-tetrazol-5-yl)-ethylam...)
Affinity DataIC50: 520nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084904(3-Dibenzofuran-3-yl-2-[1-phosphono-3-(2,3,4-trimet...)
Affinity DataIC50: 520nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084904(3-Dibenzofuran-3-yl-2-[1-phosphono-3-(2,3,4-trimet...)
Affinity DataIC50: 520nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50251742((S)-2-{(R)-2-[Hydroxy-((2R,3R,4R,5R,6S)-3,4,5-trih...)
Affinity DataIC50: 1.20E+3nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084913(2-[3-Dibenzofuran-3-yl-2-(phosphonomethyl-amino)-p...)
Affinity DataIC50: 1.64E+3nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084907(3-Dibenzofuran-3-yl-2-(3-naphthalen-1-yl-1-phospho...)
Affinity DataIC50: 1.80E+3nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084907(3-Dibenzofuran-3-yl-2-(3-naphthalen-1-yl-1-phospho...)
Affinity DataIC50: 1.80E+3nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084893(3-Dibenzofuran-3-yl-2-(phosphonomethyl-amino)-prop...)
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084909({[2-(9-Methyl-9H-carbazol-2-yl)-1-(1H-tetrazol-5-y...)
Affinity DataIC50: 4.00E+3nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50064110(CHEMBL147847 | 2-{2-[(S)-5-(2,4-Difluoro-phenyl)-2...)
Affinity DataIC50: 5.80E+3nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50084894(3-Dibenzofuran-3-yl-2-[3-(2,3-dimethoxy-phenyl)-1-...)
Affinity DataIC50: 6.40E+3nMAssay Description:In vitro inhibition of rat neutral endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
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