Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50009497
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084227(2-Diethylamino-5-methyl-4-oxo-4H-thieno[2,3-d][1,3...)
Affinity DataKd:  620nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084228(2-(diethylamino)-5-methyl-4H-thieno[2,3-d][1,3]oxa...)
Affinity DataKd:  5.50E+3nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084235(2-Diethylamino-benzo[4,5]thieno[2,3-d][1,3]oxazin-...)
Affinity DataKi:  5.80nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50064308(2-Diethylamino-5,6,7,8-tetrahydro-benzo[4,5]thieno...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084233(2-Diethylamino-6,7-dihydro-5H-cyclopenta[4,5]thien...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084232(2-Diethylamino-5-isopropyl-thieno[2,3-d][1,3]oxazi...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084234(2-Diethylamino-6,7,8,9-tetrahydro-5H-3-oxa-10-thia...)
Affinity DataKi:  44nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084227(2-Diethylamino-5-methyl-4-oxo-4H-thieno[2,3-d][1,3...)
Affinity DataKi:  91nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084230(2-Diethylamino-thieno[3,2-d][1,3]oxazin-4-one | CH...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084229(2-Diethylamino-5-methyl-5,6,7,8-tetrahydro-benzo[4...)
Affinity DataKi:  210nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084236(2-Diethylamino-thieno[2,3-d][1,3]oxazin-4-one | CH...)
Affinity DataKi:  260nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084231(2-Diethylamino-benzo[d][1,3]oxazin-4-one | CHEMBL3...)
Affinity DataKi:  310nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084228(2-(diethylamino)-5-methyl-4H-thieno[2,3-d][1,3]oxa...)
Affinity DataKi:  450nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed