Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50036766
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50082524(2,6-Bis(3-pyrrolidinopropionamido)anthracene-9,10-...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080847(N,N'-(acridine-3,6-diyl)bis(3-(piperidin-1-yl)prop...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080840(N,N'-(acridine-3,6-diyl)bis(3-(azepan-1-yl)propana...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50082532(2,6-Bis(3-piperidinopropionamido)anthracene-9,10-d...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080849(3-PYRROLIDIN-1-YL-N-[6-(3-PYRROLIDIN-1-YL-PROPIONY...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50082530(2,6-Bis[3-(hexamethyleneimino)propionamido]anthrac...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080846(3,6-Bis[3-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octa...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50082526(2,6-Bis[3-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octa...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50082528(2,6-Bis[3-(heptamethyleneimino)propionamido]anthra...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080852(3-Azocan-1-yl-N-[6-(3-azocan-1-yl-propionylamino)-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Telomerase evaluated by TRAP Assay studies.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed