Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50003524
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472306(CHEMBL93845)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  11.7nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472306(CHEMBL93845)
Affinity DataKi:  23nMAssay Description:Predicted affinity for imidazoline receptor I2 by three field CoMFA modelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50472306(CHEMBL93845)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-clonidine from Alpha-2 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]-clonidine from Alpha-2 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  251nMAssay Description:Predicted affinity for imidazoline receptor I2 by three field CoMFA modelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472307(CHEMBL2367778)
Affinity DataKi:  331nMAssay Description:Predicted affinity for imidazoline receptor I2 by three field CoMFA modelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472306(CHEMBL93845)
Affinity DataKi:  347nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472304(CHEMBL2367779)
Affinity DataKi:  724nMAssay Description:Predicted affinity for imidazoline receptor I2 by three field CoMFA modelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  891nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  891nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  5.50E+3nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  5.75E+3nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  5.75E+3nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  1.41E+4nMAssay Description:Displacement of [3H]-clonidine from Alpha-2 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  2.95E+4nMAssay Description:Displacement of [3H]-clonidine from Alpha-2 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  2.95E+4nMAssay Description:Displacement of [3H]-clonidine from Alpha-2 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed