Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50008943
LigandPNGBDBM50078723((S)-2-[(4-tert-Butyl-benzyl)-methyl-amino]-4-methy...)
Affinity DataIC50: 40nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50078730((S)-2-[(4-tert-Butyl-benzyl)-methyl-amino]-4-methy...)
Affinity DataIC50: 90nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078727((S)-2-(Cyclohexyl-methyl-amino)-4-methyl-pentanoic...)
Affinity DataIC50: 200nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078724((S)-2-[(4-tert-Butyl-benzyl)-methyl-amino]-4-methy...)
Affinity DataIC50: 270nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078745((S)-2-[(4-tert-Butyl-benzyl)-methyl-amino]-4-methy...)
Affinity DataIC50: 310nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078743((S)-2-(Cyclohexylmethyl-methyl-amino)-4-methyl-pen...)
Affinity DataIC50: 310nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078725((S)-4-Methyl-2-[methyl-(3-methyl-butyl)-amino]-pen...)
Affinity DataIC50: 320nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078740((S)-2-(Cyclohexylmethyl-methyl-amino)-4-methyl-pen...)
Affinity DataIC50: 320nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078744((S)-2-(Cyclohexyl-methyl-amino)-4-methyl-pentanoic...)
Affinity DataIC50: 380nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078742((S)-2-(Cyclohexylmethyl-methyl-amino)-4-methyl-pen...)
Affinity DataIC50: 420nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078735((S)-2-[(4-tert-Butyl-benzyl)-methyl-amino]-4-methy...)
Affinity DataIC50: 440nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078729((S)-2-[(4-tert-Butyl-benzyl)-methyl-amino]-4-methy...)
Affinity DataIC50: 500nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078718((S)-2-(Cyclohexylmethyl-methyl-amino)-4-methyl-pen...)
Affinity DataIC50: 500nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078739((S)-4-Methyl-2-[methyl-(3-methyl-butyl)-amino]-pen...)
Affinity DataIC50: 590nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078746((S)-4-Methyl-2-[methyl-(3-methyl-butyl)-amino]-pen...)
Affinity DataIC50: 660nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078736((S)-2-(Cyclohexyl-methyl-amino)-4-methyl-pentanoic...)
Affinity DataIC50: 760nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078732((S)-2-(Cyclohexyl-methyl-amino)-4-methyl-pentanoic...)
Affinity DataIC50: 880nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078741((S)-4-Methyl-2-[methyl-(3-methyl-butyl)-amino]-pen...)
Affinity DataIC50: 880nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078726((S)-2-(Cyclohexylmethyl-methyl-amino)-4-methyl-pen...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078731((S)-4-Methyl-2-[methyl-(3-methyl-butyl)-amino]-pen...)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078728((S)-2-Dimethylamino-4-methyl-pentanoic acid [(S)-1...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078719((S)-2-(Cyclohexylmethyl-methyl-amino)-4-methyl-pen...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078738((S)-4-Methyl-2-[methyl-(3-methyl-butyl)-amino]-pen...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078721((S)-2-(Cyclohexyl-methyl-amino)-4-methyl-pentanoic...)
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078737((S)-2-Dimethylamino-4-methyl-pentanoic acid [(S)-1...)
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078722((S)-2-Dimethylamino-4-methyl-pentanoic acid [(S)-2...)
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078720((S)-2-Dimethylamino-4-methyl-pentanoic acid [(S)-2...)
Affinity DataIC50: 2.80E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078734((S)-2-Dimethylamino-4-methyl-pentanoic acid [(S)-2...)
Affinity DataIC50: 4.10E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078717((S)-2-(Cyclohexyl-methyl-amino)-4-methyl-pentanoic...)
Affinity DataIC50: 5.60E+3nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50078733((S)-2-Dimethylamino-4-methyl-pentanoic acid [(S)-1...)
Affinity DataIC50: 1.30E+4nMAssay Description:In vitro antagonism of N-type voltage sensitive calcium channel in IMR-32 assay using fluorescent [Ca2+] indicator Indo-11 in the presence of 5 uM ni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed