Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50008831
Affinity DataKi: 2.60nMAssay Description:In vitro binding affinity against 5-HT1A receptor of rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:In vitro binding affinity against 5-HT1A receptor of rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:In vitro binding affinity against 5-HT1A receptor of rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rat)
Postech
Curated by ChEMBL
Postech
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:In vitro binding affinity against Alpha-2 adrenergic receptor of rat cerebral cortex using [3H]RX-821002More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rat)
Postech
Curated by ChEMBL
Postech
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:In vitro binding affinity against Alpha-2 adrenergic receptor of rat cerebral cortex using [3H]RX-821002More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:In vitro binding affinity against 5-HT1A receptor of rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:In vitro binding affinity against 5-HT1A receptor of rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rat)
Postech
Curated by ChEMBL
Postech
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:In vitro binding affinity against Alpha-2 adrenergic receptor of rat cerebral cortex using [3H]RX-821002More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rat)
Postech
Curated by ChEMBL
Postech
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:In vitro binding affinity against Alpha-2 adrenergic receptor of rat cerebral cortex using [3H]RX-821002More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vitro binding affinity against 5-HT1A receptor of rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:In vitro binding affinity against 5-HT1A receptor of rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:In vitro binding affinity against 5-HT2A receptor of rat cerebral cortex using [3H]ketanserinMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rat)
Postech
Curated by ChEMBL
Postech
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:In vitro binding affinity against Alpha-2 adrenergic receptor of rat cerebral cortex using [3H]RX-821002More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:In vitro binding affinity against 5-HT2A receptor of rat cerebral cortex using [3H]ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:In vitro binding affinity against 5-HT2A receptor of rat cerebral cortex using [3H]ketanserinMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rat)
Postech
Curated by ChEMBL
Postech
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:In vitro binding affinity against Alpha-2 adrenergic receptor of rat cerebral cortex using [3H]RX-821002More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:In vitro binding affinity against Dopamine receptor D2 of rat striatum using [3H]racloprideMore data for this Ligand-Target Pair
Affinity DataKi: 184nMAssay Description:In vitro binding affinity against 5-HT2A receptor of rat cerebral cortex using [3H]ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: 185nMAssay Description:In vitro binding affinity against Dopamine receptor D2 of rat striatum using [3H]racloprideMore data for this Ligand-Target Pair
Affinity DataKi: 195nMAssay Description:In vitro binding affinity against Dopamine receptor D2 of rat striatum using [3H]racloprideMore data for this Ligand-Target Pair
Affinity DataKi: 232nMAssay Description:In vitro binding affinity against 5-HT2A receptor of rat cerebral cortex using [3H]ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: 263nMAssay Description:In vitro binding affinity against Dopamine receptor D2 of rat striatum using [3H]racloprideMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:In vitro binding affinity against 5-HT2A receptor of rat cerebral cortex using [3H]ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: 327nMAssay Description:In vitro binding affinity against Dopamine receptor D2 of rat striatum using [3H]racloprideMore data for this Ligand-Target Pair
Affinity DataKi: 334nMAssay Description:In vitro binding affinity against Dopamine receptor D2 of rat striatum using [3H]racloprideMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rat)
Postech
Curated by ChEMBL
Postech
Curated by ChEMBL
Affinity DataKi: 334nMAssay Description:In vitro binding affinity against Alpha-2 adrenergic receptor of rat cerebral cortex using [3H]RX-821002More data for this Ligand-Target Pair
Affinity DataKi: >367nMAssay Description:In vitro binding affinity against 5-HT2A receptor of rat cerebral cortex using [3H]ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: 783nMAssay Description:In vitro binding affinity against Dopamine receptor D2 of rat striatum using [3H]racloprideMore data for this Ligand-Target Pair
Affinity DataKi: 1.57E+3nMAssay Description:In vitro binding affinity against Dopamine receptor D1 of rat striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:In vitro binding affinity against Dopamine receptor D1 of rat striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:In vitro binding affinity against Dopamine receptor D1 of rat striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataKi: 6.67E+3nMAssay Description:In vitro binding affinity against Dopamine receptor D1 of rat striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataKi: 1.25E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D1 of rat striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataKi: 3.76E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D1 of rat striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataKi: 8.81E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D1 of rat striatum using [3H]SCH-23390More data for this Ligand-Target Pair
