Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50008759
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076903(3-(2-Bromo-4-isopropyl-phenyl)-7-(cyclopropylmethy...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076905(3-(2-Bromo-4-isopropyl-phenyl)-7-diethylamino-5-me...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076902(7-[Bis-(2-methoxy-ethyl)-amino]-5-methyl-3-(2,4,6-...)
Affinity DataKi:  5nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076899(7-[Bis-(2-methoxy-ethyl)-amino]-3-(2-bromo-4-isopr...)
Affinity DataKi:  6.60nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076906(7-[Bis-(2-methoxy-ethyl)-amino]-5-methyl-3-(2,4,6-...)
Affinity DataKi:  8.60nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076901(7-Diethylamino-5-methyl-3-(2,4,6-trimethyl-phenyl)...)
Affinity DataKi:  9.20nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076900(3-(2-Bromo-4-isopropyl-phenyl)-7-diethylamino-5-me...)
Affinity DataKi:  9.40nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076893(3-(2-Bromo-4-isopropyl-phenyl)-7-(cyclopropylmethy...)
Affinity DataKi:  13nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076897(7-(Cyclopropylmethyl-propyl-amino)-5-methyl-3-(2,4...)
Affinity DataKi:  13nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076892(7-Diethylamino-5-methyl-3-(2,4,6-trimethyl-phenyl)...)
Affinity DataKi:  15nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076894(7-[Bis-(2-methoxy-ethyl)-amino]-3-(2-bromo-4-isopr...)
Affinity DataKi:  15nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076898(7-(Cyclopropylmethyl-propyl-amino)-5-methyl-3-(2,4...)
Affinity DataKi:  16nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076896(3-(2-Bromo-4-isopropyl-phenyl)-7-(butyl-ethyl-amin...)
Affinity DataKi:  24nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076904(3-(2-Bromo-4-isopropyl-phenyl)-7-(di-sec-butyl-ami...)
Affinity DataKi:  45nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076895(3-(2-Bromo-4-isopropyl-phenyl)-5-methyl-7-morpholi...)
Affinity DataKi:  122nMAssay Description:Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed