Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50008746
LigandPNGBDBM50076802(Lithium; (S)-2-{[2'-methyl-5-(5-pyridin-4-yl-furan...)
Affinity DataEC50: >0.300nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076806(Lithium; (S)-2-({5-[5-(4-methoxy-phenyl)-furan-2-y...)
Affinity DataEC50: >1nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076801(Lithium; (S)-2-({2'-methyl-5-[5-(3-nitro-phenyl)-f...)
Affinity DataEC50:  10nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076803(Lithium; (S)-2-({5-[5-(2-fluoro-phenyl)-furan-2-yl...)
Affinity DataEC50: >1nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076794(Lithium; (S)-2-({5-[5-(4-isopropyl-phenyl)-furan-2...)
Affinity DataEC50:  0.780nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076797(Lithium; (S)-2-{[2'-methyl-5-(5-phenyl-furan-2-ylm...)
Affinity DataEC50: >1nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076809(Lithium; (S)-2-({5-[5-(4-formyl-phenyl)-furan-2-yl...)
Affinity DataEC50: >1nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076791(Lithium; (S)-4-methylsulfanyl-2-{[2'-methyl-5-(5-p...)
Affinity DataEC50:  1.80nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076793(Lithium; (S)-2-({2'-methyl-5-[5-(4-methylsulfanyl-...)
Affinity DataEC50:  10nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076800(Lithium; (S)-2-({5-[5-(4-acetyl-phenyl)-furan-2-yl...)
Affinity DataEC50: >1nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076795(Lithium; (S)-2-({5-[5-(4-dimethylamino-phenyl)-fur...)
Affinity DataEC50:  0.900nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076788(Lithium; (S)-2-({5-[5-(3-fluoro-phenyl)-furan-2-yl...)
Affinity DataEC50:  10nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076811(Lithium; (S)-2-({5-[5-(4-chloro-phenyl)-furan-2-yl...)
Affinity DataEC50:  0.100nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076810(Lithium; (S)-4-methylsulfanyl-2-({2'-methyl-5-[5-(...)
Affinity DataEC50:  1.20nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076808(Lithium; (S)-2-{[2'-methyl-5-(5-pyridin-2-yl-furan...)
Affinity DataEC50: >0.300nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076807(Lithium; (S)-2-({5-[5-(3-methoxy-phenyl)-furan-2-y...)
Affinity DataEC50: >1nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076790(Lithium; (S)-2-{[2'-methyl-5-(5-pyridin-3-yl-furan...)
Affinity DataEC50:  0.300nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076813(Lithium; (S)-2-({5-[5-(2-methoxy-phenyl)-furan-2-y...)
Affinity DataEC50: >1nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076798(Lithium; (S)-2-({5-[5-(4-fluoro-phenyl)-furan-2-yl...)
Affinity DataEC50:  1.5nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50067563((S)-2-{[2'-Methyl-5-(pyridin-3-yloxymethyl)-biphen...)
Affinity DataIC50: 0.400nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50067584(2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bipheny...)
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076811(Lithium; (S)-2-({5-[5-(4-chloro-phenyl)-furan-2-yl...)
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076809(Lithium; (S)-2-({5-[5-(4-formyl-phenyl)-furan-2-yl...)
Affinity DataIC50: 1.20nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076798(Lithium; (S)-2-({5-[5-(4-fluoro-phenyl)-furan-2-yl...)
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076802(Lithium; (S)-2-{[2'-methyl-5-(5-pyridin-4-yl-furan...)
Affinity DataIC50: 2.40nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076795(Lithium; (S)-2-({5-[5-(4-dimethylamino-phenyl)-fur...)
Affinity DataIC50: 2.60nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076794(Lithium; (S)-2-({5-[5-(4-isopropyl-phenyl)-furan-2...)
Affinity DataIC50: 2.90nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076791(Lithium; (S)-4-methylsulfanyl-2-{[2'-methyl-5-(5-p...)
Affinity DataIC50: 2.90nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076810(Lithium; (S)-4-methylsulfanyl-2-({2'-methyl-5-[5-(...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076799((S)-2-{[5-(5-Bromo-furan-2-ylmethoxymethyl)-2'-met...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076792(Lithium; (S)-2-({5-[5-(4-chloro-3-fluoro-phenyl)-f...)
Affinity DataIC50: 4.90nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076801(Lithium; (S)-2-({2'-methyl-5-[5-(3-nitro-phenyl)-f...)
Affinity DataIC50: 6nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076797(Lithium; (S)-2-{[2'-methyl-5-(5-phenyl-furan-2-ylm...)
Affinity DataIC50: 6nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076793(Lithium; (S)-2-({2'-methyl-5-[5-(4-methylsulfanyl-...)
Affinity DataIC50: 6.20nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076803(Lithium; (S)-2-({5-[5-(2-fluoro-phenyl)-furan-2-yl...)
Affinity DataIC50: 6.30nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076790(Lithium; (S)-2-{[2'-methyl-5-(5-pyridin-3-yl-furan...)
Affinity DataIC50: 6.5nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076800(Lithium; (S)-2-({5-[5-(4-acetyl-phenyl)-furan-2-yl...)
Affinity DataIC50: 6.60nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076788(Lithium; (S)-2-({5-[5-(3-fluoro-phenyl)-furan-2-yl...)
Affinity DataIC50: 7.60nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076806(Lithium; (S)-2-({5-[5-(4-methoxy-phenyl)-furan-2-y...)
Affinity DataIC50: 8.40nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076804(Lithium; (S)-4-methylsulfanyl-2-({2'-methyl-5-[5-(...)
Affinity DataIC50: 8.80nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076789(Lithium; (S)-4-methylsulfanyl-2-({2'-methyl-5-[5-(...)
Affinity DataIC50: 9.90nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076807(Lithium; (S)-2-({5-[5-(3-methoxy-phenyl)-furan-2-y...)
Affinity DataIC50: 12nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076808(Lithium; (S)-2-{[2'-methyl-5-(5-pyridin-2-yl-furan...)
Affinity DataIC50: 19nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076813(Lithium; (S)-2-({5-[5-(2-methoxy-phenyl)-furan-2-y...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076812((S)-2-[(5-{[(Furan-2-ylmethyl)-amino]-methyl}-biph...)
Affinity DataIC50: 560nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50076805((S)-4-Methylsulfanyl-2-[(5-phenoxymethyl-biphenyl-...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory activity was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed