Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50035038
TargetProthrombin(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50075822(ORG-37476 | N-[1-(1-Amino-isoquinolin-6-ylmethyl)-...)
Affinity DataIC50: 82nMAssay Description:Compound was tested for inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50037996(N-[1-(4-Carbamimidoyl-benzyl)-2-oxo-2-piperidin-1-...)
Affinity DataIC50: 169nMAssay Description:Compound was tested for inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50037996(N-[1-(4-Carbamimidoyl-benzyl)-2-oxo-2-piperidin-1-...)
Affinity DataIC50: 690nMAssay Description:Compound was tested for inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50075824(Aminoisoquinoline derivative | CHEMBL351865)
Affinity DataIC50: 1.10E+3nMAssay Description:Compound was tested for inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50075826(N-[1-(1-Amino-isoquinolin-6-ylmethyl)-2-oxo-2-pipe...)
Affinity DataIC50: 2.80E+4nMAssay Description:Compound was tested for inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50075823(N-[1-(1-Amino-isoquinolin-6-ylmethyl)-2-oxo-2-pipe...)
Affinity DataIC50: 5.50E+4nMAssay Description:Compound was tested for inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50075823(N-[1-(1-Amino-isoquinolin-6-ylmethyl)-2-oxo-2-pipe...)
Affinity DataIC50: 2.55E+5nMAssay Description:Compound was tested for inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50075825(N-[1-(1-Amino-isoquinolin-6-ylmethyl)-2-oxo-2-pipe...)
Affinity DataIC50: 3.57E+5nMAssay Description:Compound was tested for inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine protease 1(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50075822(ORG-37476 | N-[1-(1-Amino-isoquinolin-6-ylmethyl)-...)
Affinity DataIC50: 3.78E+5nMAssay Description:Compound was tested for inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed