Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50008628
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075421(7-(Ethyl-methanesulfonyl-amino)-1-(2-methoxy-benzy...)
Affinity DataIC50: 3.60nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075429(7-(Methanesulfonyl-methyl-amino)-1-(2-methoxy-benz...)
Affinity DataIC50: 8.60nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075422(7-(Methanesulfonyl-propyl-amino)-1-(2-methoxy-benz...)
Affinity DataIC50: 13nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075412(1-(2,5-Dimethoxy-benzyl)-4-(4-methoxy-phenyl)-2-ox...)
Affinity DataIC50: 21nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075435(7-Amino-1-(2-methoxy-benzyl)-4-(4-methoxy-phenyl)-...)
Affinity DataIC50: 27nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075412(1-(2,5-Dimethoxy-benzyl)-4-(4-methoxy-phenyl)-2-ox...)
Affinity DataIC50: 41nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075424(7-Methanesulfonylamino-1-(2-methoxy-benzyl)-4-(4-m...)
Affinity DataIC50: 120nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075417(1-(2-Methoxy-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,...)
Affinity DataIC50: 120nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075428(1-(2-Methoxy-benzyl)-2-oxo-4-(3,4,5-trimethoxy-phe...)
Affinity DataIC50: 170nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075419(1-(2-Methoxy-benzyl)-4-(4-methoxy-phenyl)-7-nitro-...)
Affinity DataIC50: 200nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075413(4-(4-Methoxy-phenyl)-1-(2-methyl-benzyl)-2-oxo-1,2...)
Affinity DataIC50: 300nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075417(1-(2-Methoxy-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,...)
Affinity DataIC50: 380nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075413(4-(4-Methoxy-phenyl)-1-(2-methyl-benzyl)-2-oxo-1,2...)
Affinity DataIC50: 420nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075415(4-(2,4-Dimethoxy-phenyl)-1-(2-methoxy-benzyl)-2-ox...)
Affinity DataIC50: 430nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075420(4-(2,5-Dimethoxy-phenyl)-1-(2-methoxy-benzyl)-2-ox...)
Affinity DataIC50: 490nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075416(1-(2-Isopropyl-benzyl)-4-(4-methoxy-phenyl)-2-oxo-...)
Affinity DataIC50: 660nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075416(1-(2-Isopropyl-benzyl)-4-(4-methoxy-phenyl)-2-oxo-...)
Affinity DataIC50: 710nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075418(1-(2-Ethoxy-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,2...)
Affinity DataIC50: 900nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075426(4-Benzo[1,3]dioxol-5-yl-1-(2-methoxy-benzyl)-2-oxo...)
Affinity DataIC50: 1.20E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075415(4-(2,4-Dimethoxy-phenyl)-1-(2-methoxy-benzyl)-2-ox...)
Affinity DataIC50: 1.20E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075411(1-(2-Chloro-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,2...)
Affinity DataIC50: 1.30E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075418(1-(2-Ethoxy-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,2...)
Affinity DataIC50: 1.30E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075433(1-(2-Methoxy-benzyl)-4-(3-methoxy-phenyl)-2-oxo-1,...)
Affinity DataIC50: 1.50E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075434(1-(3-Methoxy-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,...)
Affinity DataIC50: 1.60E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075426(4-Benzo[1,3]dioxol-5-yl-1-(2-methoxy-benzyl)-2-oxo...)
Affinity DataIC50: 1.90E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075419(1-(2-Methoxy-benzyl)-4-(4-methoxy-phenyl)-7-nitro-...)
Affinity DataIC50: 2.10E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075435(7-Amino-1-(2-methoxy-benzyl)-4-(4-methoxy-phenyl)-...)
Affinity DataIC50: 2.30E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075411(1-(2-Chloro-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,2...)
Affinity DataIC50: 2.70E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075427(1-Benzyl-4-(4-methoxy-phenyl)-2-oxo-1,2-dihydro-be...)
Affinity DataIC50: 2.70E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075430(4-(4-Methoxy-phenyl)-1-(2-methylsulfanyl-benzyl)-2...)
Affinity DataIC50: 2.70E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075434(1-(3-Methoxy-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,...)
Affinity DataIC50: 2.70E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075427(1-Benzyl-4-(4-methoxy-phenyl)-2-oxo-1,2-dihydro-be...)
Affinity DataIC50: 3.00E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075433(1-(2-Methoxy-benzyl)-4-(3-methoxy-phenyl)-2-oxo-1,...)
Affinity DataIC50: 3.50E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075425(1-(2,3-Dimethoxy-benzyl)-4-(4-methoxy-phenyl)-2-ox...)
Affinity DataIC50: 3.50E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075425(1-(2,3-Dimethoxy-benzyl)-4-(4-methoxy-phenyl)-2-ox...)
Affinity DataIC50: 5.20E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075430(4-(4-Methoxy-phenyl)-1-(2-methylsulfanyl-benzyl)-2...)
Affinity DataIC50: 6.40E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075420(4-(2,5-Dimethoxy-phenyl)-1-(2-methoxy-benzyl)-2-ox...)
Affinity DataIC50: 6.80E+3nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075421(7-(Ethyl-methanesulfonyl-amino)-1-(2-methoxy-benzy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075436(1-(2,6-Dimethoxy-benzyl)-4-(4-methoxy-phenyl)-2-ox...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075431(1-(4-Methoxy-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075423(1-(2-Methoxy-benzyl)-4-(2-methoxy-phenyl)-2-oxo-1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075414(1-Benzyl-2-oxo-4-phenyl-1,2-dihydro-benzo[4,5]furo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075432(4-(4-Methoxy-phenyl)-2-oxo-1-(2,4,5-trimethoxy-ben...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075422(7-(Methanesulfonyl-propyl-amino)-1-(2-methoxy-benz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075436(1-(2,6-Dimethoxy-benzyl)-4-(4-methoxy-phenyl)-2-ox...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075429(7-(Methanesulfonyl-methyl-amino)-1-(2-methoxy-benz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075424(7-Methanesulfonylamino-1-(2-methoxy-benzyl)-4-(4-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075423(1-(2-Methoxy-benzyl)-4-(2-methoxy-phenyl)-2-oxo-1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-1 receptor(Rat)
Merck

Curated by ChEMBL
LigandPNGBDBM50075432(4-(4-Methoxy-phenyl)-2-oxo-1-(2,4,5-trimethoxy-ben...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin A receptor in rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50075431(1-(4-Methoxy-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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