Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50008567
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074768(2-{2-[Bis-(4-methoxycarbonyl-phenoxy)-phosphoryl]-...)
Affinity DataIC50: 16nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074760(2-(2-{Bis-[4-(ethoxycarbonylmethyl-carbamoyl)-phen...)
Affinity DataIC50: 23nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074762(2-{2-[Bis-(4-propylcarbamoyl-phenoxy)-phosphoryl]-...)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074769(2-(2-{Bis-[4-(2-methoxycarbonyl-ethylcarbamoyl)-ph...)
Affinity DataIC50: 36nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074753(2-{2-[Bis-(4-methanesulfonylamino-phenoxy)-phospho...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074766(2-{2-[Bis-(4-acetylamino-phenoxy)-phosphoryl]-pyrr...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074759(2-(2-{Bis-[4-(2-amino-acetylamino)-phenoxy]-phosph...)
Affinity DataIC50: 500nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074770(2-(2-{[4-((R)-2-Amino-propionylamino)-phenoxy]-[4-...)
Affinity DataIC50: 600nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074772(2-(2-{Bis-[4-(2-benzoylamino-acetylamino)-phenoxy]...)
Affinity DataIC50: 700nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074756(2-{2-[Bis-(3-acetylamino-phenoxy)-phosphoryl]-pyrr...)
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074767(2-(2-{Bis-[4-(2-acetylamino-2-methoxycarbonyl-ethy...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074765(2-{2-[(5-Ureido-cyclohexa-1,3-dienyloxy)-(3-ureido...)
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074752(2-(2-{Bis-[4-(pyrrolidin-1-ylamino)-phenoxy]-phosp...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074761((R)-2-[2-(Diphenoxy-phosphoryl)-pyrrolidine-1-carb...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074758((S)-2-[2-(Diphenoxy-phosphoryl)-pyrrolidine-1-carb...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074757(2-{2-[Bis-(4-methoxy-phenoxy)-phosphoryl]-pyrrolid...)
Affinity DataIC50: 2.20E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074751((S)-2-[2-(6-Oxo-5,7-dioxa-6lambda*5*-phospha-diben...)
Affinity DataIC50: 3.10E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074764((S)-2-{2-[(2'-Hydroxy-biphenyl-2-yloxy)-methoxy-ph...)
Affinity DataIC50: 4.70E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074756(2-{2-[Bis-(3-acetylamino-phenoxy)-phosphoryl]-pyrr...)
Affinity DataIC50: 5.00E+4nMAssay Description:Effect on the activity of prolyl endopeptidase (PEP) was evaluated at 1 mM concentration for DPP IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074761((R)-2-[2-(Diphenoxy-phosphoryl)-pyrrolidine-1-carb...)
Affinity DataIC50: 8.30E+4nMAssay Description:Effect on the activity of membrane alanyl aminopeptidase (MAAP) is evaluated at at a concentration of 1 mM.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074756(2-{2-[Bis-(3-acetylamino-phenoxy)-phosphoryl]-pyrr...)
Affinity DataIC50: 8.90E+4nMAssay Description:Effect on the activity of prolyl endopeptidase (PEP) was evaluated at the IC50 concentration for DPP IV andMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074760(2-(2-{Bis-[4-(ethoxycarbonylmethyl-carbamoyl)-phen...)
Affinity DataIC50: 1.04E+5nMAssay Description:Effect on the activity of membrane alanyl aminopeptidase (MAAP) is evaluated at the IC50 concentration for DPPIV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074754(2-{2-[Bis-(4-hydroxy-phenoxy)-phosphoryl]-pyrrolid...)
Affinity DataIC50: 1.90E+5nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074763(2-{2-[Bis-(2,2,2-trichloro-ethoxy)-phosphoryl]-pyr...)
Affinity DataIC50: 1.80E+6nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074755(2-{2-[Bis-(2,2,2-trifluoro-ethoxy)-phosphoryl]-pyr...)
Affinity DataIC50: 9.10E+6nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed