Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50003538
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403759(CHEMBL428494)
Affinity DataKi:  1.90nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi:  2.10nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403770(CHEMBL12427)
Affinity DataKi:  3.30nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403768(CHEMBL273246)
Affinity DataKi:  3.80nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403777(CHEMBL12702)
Affinity DataKi:  5.10nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50130272(2a-[3-(4-Phenyl-piperazin-1-yl)-propyl]-2a,3,4,5-t...)
Affinity DataKi:  5.20nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403772(CHEMBL268921)
Affinity DataKi:  5.40nMAssay Description:Compound was evaluated for its ability to displace [3H]ketanserin binding from cloned rat cerebral cortex membranes 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50130272(2a-[3-(4-Phenyl-piperazin-1-yl)-propyl]-2a,3,4,5-t...)
Affinity DataKi:  16nMAssay Description:Compound was evaluated for its ability to displace [3H]ketanserin binding from cloned rat cerebral cortex membranes 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403770(CHEMBL12427)
Affinity DataKi:  43nMAssay Description:Compound was evaluated for its ability to displace [3H]ketanserin binding from cloned rat cerebral cortex membranes 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403759(CHEMBL428494)
Affinity DataKi:  54nMAssay Description:Compound was evaluated for its ability to displace [3H]ketanserin binding from cloned rat cerebral cortex membranes 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi:  98nMAssay Description:Compound was evaluated for its ability to displace [3H]ketanserin binding from cloned rat cerebral cortex membranes 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403772(CHEMBL268921)
Affinity DataKi:  102nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi:  105nMAssay Description:Compound was evaluated for its ability to displace [3H]spiperone binding from Dopamine receptor D2 in rat striatum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403768(CHEMBL273246)
Affinity DataKi:  105nMAssay Description:Compound was evaluated for its ability to displace [3H]ketanserin binding from cloned rat cerebral cortex membranes 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403777(CHEMBL12702)
Affinity DataKi:  112nMAssay Description:Compound was evaluated for its ability to displace [3H]ketanserin binding from cloned rat cerebral cortex membranes 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi:  170nMAssay Description:Compound was evaluated for its ability to displace [3H]8-OH-DPAT binding from human 5-hydroxytryptamine 1A receptor in mammalian cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi:  525nMAssay Description:Compound was evaluated for its ability to displace [3H]LSD binding from human recombinant 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi: <1.00E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]GR-113808 binding from 5-hydroxytryptamine 4 receptor in guinea pig striatum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403783(CHEMBL273890)
Affinity DataKi: <1.00E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403783(CHEMBL273890)
Affinity DataKi: <1.00E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]ketanserin binding from cloned rat cerebral cortex membranes 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed