Compile Data Set for Download or QSAR
Report error Found 21 of ic50 data for polymerid = 8889,8891,50001840
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50535485(CHEMBL4594145)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of VKOR (unknown origin) in HEK293 expressing FIXgla-PC incubated for 48 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50343352(2-hydroxy-3-(3-oxo-1-phenylbutyl)-4H-chromen-4-one...)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of VKOR (unknown origin) in HEK293 expressing FIXgla-PC incubated for 48 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50166637(2'-Biphenyl-4-yl-4-hydroxy-3',4'-dihydro-2'H-[3,4'...)
Affinity DataIC50: 40nMAssay Description:Inhibitory concentration against beef liver Vitamin K epoxide reductase (vitamin K 2,3-epoxide reductase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50535487(CHEMBL4530669)
Affinity DataIC50: 58nMAssay Description:Inhibition of VKOR (unknown origin) in HEK293 expressing FIXgla-PC incubated for 48 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50535484(CHEMBL4517532)
Affinity DataIC50: 59nMAssay Description:Inhibition of VKOR (unknown origin) in HEK293 expressing FIXgla-PC incubated for 48 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50535488(CHEMBL4443961)
Affinity DataIC50: 90nMAssay Description:Inhibition of VKOR (unknown origin) in HEK293 expressing FIXgla-PC incubated for 48 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629252(CHEMBL5435296)
Affinity DataIC50: 98nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629253(CHEBI:81892 | Brodifacoum | BRODIFACOUM)
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629247(CHEMBL5436380)
Affinity DataIC50: 498nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629246(CHEMBL5433796)
Affinity DataIC50: 527nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629245(CHEMBL5432023)
Affinity DataIC50: 643nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629250(CHEMBL5403819)
Affinity DataIC50: 873nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50166638(13-(4-phenylphenyl)-4,12,14-trioxapentacyclo[11.7....)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against beef liver Vitamin K epoxide reductase (vitamin K 2,3-epoxide reductase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50343352(2-hydroxy-3-(3-oxo-1-phenylbutyl)-4H-chromen-4-one...)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629244(CHEMBL5404461)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50535486(CHEMBL4463800)
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of VKOR (unknown origin) in HEK293 expressing FIXgla-PC incubated for 48 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629248(CHEMBL5434421)
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629249(CHEMBL5396437)
Affinity DataIC50: 5.54E+3nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629254(Warfarin alcohol | WARFARIN ALCOHOL)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629251(CHEMBL5424000)
Affinity DataIC50: 2.39E+4nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50629255(Isoprenylcoumarin | ISOPRENYLCOUMARIN)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed