Compile Data Set for Download or QSAR
Report error Found 3419 of ic50 data for polymerid = 704,751,752,753,754,771,772,778,966,1307,6607,10075,10147,50001106,50004392,50004401
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50181441(CHEBI:85202 | BCX-1812 | Peramivir)
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of influenza virus neuraminidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5258/2009(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50401401(CHEMBL2206459)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Influenza A virus (A/reassortant/NIBRG-14(Viet Nam/1194/2004 x Puerto Rico/8/1934)(H5N1)) neuraminidase in virus-infected allantoic flu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5555/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/HH/1580/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50078329(4-[2,2-bis(hydroxymethyl)-5-oxopyrrolidin-1-yl]-3-...)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of influenza virus neuraminidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50181441(CHEBI:85202 | BCX-1812 | Peramivir)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of oseltamivir-resistant Influenza A virus A/WSN/1933(H1N1) recombinant wild type neuraminidase transfected in HEK293 cells using MUNANA a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50401401(CHEMBL2206459)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of wild type Influenza A virus A/WSN/1933(H1N1) neuraminidase in virus-infected allantoic fluid using 2'-(4-methylumbelliferyl)-alpha-D-N-...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Influenza A virus (A/duck/Laos/25/2006(H5N1)) neuraminidase isolated from virus-infected BALB/c mouse by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Influenza A virus (A/duck/Laos/25/2006(H5N1)) neuraminidase by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50484773(Oseltamivir Potassium Carboxylate | OSELTAMIVIR PO...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Influenza A virus H7N3 N3 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50484774(CHEMBL1956716)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Influenza A virus H7N3 N3 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5555/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50631705(CHEMBL5415752)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of influenza A virus neuraminidaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
The Hong Kong Polytechnic University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of influenza A virus H3N2 clinical isolate neuraminidase using NA-Fluor MUNANA as substrate preincubated for 20 to 30 mins followed by sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5258/2009(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/HH/1580/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50028503(Guanidino-Oseltamivir Carboxylicacid | CHEMBL81717)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/HH/1580/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Berlin/10/04(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.170nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Rheinland-Pfalz/3911/03(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.180nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Sachsen/6/02(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50028503(Guanidino-Oseltamivir Carboxylicacid | CHEMBL81717)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5258/2009(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Influenza A virus (A/Thailand/1(KAN-1)/2004(H5N1)) neuraminidase isolated from virus-infected BALB/c mouse by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50028503(Guanidino-Oseltamivir Carboxylicacid | CHEMBL81717)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Influenza virus neuraminidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM5025(ethyl (3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-y...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Influenza A virus H7N3 N3 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM5025(ethyl (3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-y...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Influenza A virus (A/Hong Kong/1/1968(H3N2)) neuraminidase by chemiluminescence based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Rheinland-Pfalz/3911/03(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 0.290nMAssay Description:Inhibition of neuraminidase H274Y mutant in Oseltamivir-resistant Influenza A virus A/Berlin/55/08(H1N1) using Na-star as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Gilead Sciences

LigandPNGBDBM5003((3R,4R,5S)-5-amino-4-acetamido-3-{[(3S)-1-phenylpe...)
Affinity DataIC50: 0.300nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50181441(CHEBI:85202 | BCX-1812 | Peramivir)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of oseltamivir-resistant Influenza A virus A/Vietnam/1194/2004(H5N1) recombinant wild type neuraminidase transfected in HEK293 cells using...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50181444(CHEMBL3818436)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of oseltamivir-resistant Influenza A virus A/Vietnam/1194/2004(H5N1) recombinant wild type neuraminidase transfected in HEK293 cells using...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50181444(CHEMBL3818436)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of oseltamivir-resistant Influenza A virus A/WSN/1933(H1N1) recombinant wild type neuraminidase transfected in HEK293 cells using MUNANA a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Gilead Sciences

LigandPNGBDBM50097655((4S,5R,6R)-4-Amino-6-dipropylcarbamoyl-5-(2,2,2-tr...)
Affinity DataIC50: 0.300nMAssay Description:Inhibitory activity against influenza A sialidase (Aichi)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Influenza A virus (A/Thailand/1(KAN-1)/2004(H5N1)) neuraminidase by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(CHEBI:85202 | BCX-1812 | Peramivir)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase expressed in HEK293 cells pre-incubated for 10 mins before 4-M...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM5025(ethyl (3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-y...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Influenza A virus (A/Puerto Rico/8/1934(H1N1)) neuraminidase by chemiluminescence based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50496023(CHEMBL3120197)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/HH/1580/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50478617(CHEMBL460452)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of influenza virus neuraminidaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50028503(Guanidino-Oseltamivir Carboxylicacid | CHEMBL81717)
Affinity DataIC50: 0.310nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5555/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50182249(CHEMBL3818159)
Affinity DataIC50: 0.350nMAssay Description:Inhibition of Influenza A virus (A/duck/Tsukuba/28/2005(H6N2)) neuraminidase N2 activity using 4MU-Neu5Ac as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus (A/Udorn/307/1972(H3N2)))
The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50401401(CHEMBL2206459)
Affinity DataIC50: 0.350nMAssay Description:Inhibition of Influenza A virus A/Udorn/1972(H3N2) neuraminidase in virus-infected allantoic fluid using 2'-(4-methylumbelliferyl)-alpha-D-N-acetylne...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50365361(CHEMBL4161935)
Affinity DataIC50: 0.350nMAssay Description:Inhibition of Influenza A virus (A/chicken/china/415/2013(H9N2)) neuraminidase activity using 4-MUNANA as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of oseltamivir-resistant Influenza A virus A/WSN/1933(H1N1) recombinant wild type neuraminidase transfected in HEK293 cells using MUNANA a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50181441(CHEBI:85202 | BCX-1812 | Peramivir)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Influenza A virus (A/WSN/1933(H1N1)) recombinant neuraminidase expressed in HEK293 cells pre-incubated for 10 mins before 4-MUNANA subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50619652(CHEMBL5417759)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of influenza A virus neuraminidaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50464877(CHEMBL4288789)
Affinity DataIC50: 0.440nMAssay Description:Inhibition of Influenza A virus (A/WSN/1933(H1N1)) neuraminidase pre-incubated for 10 mins before 4-MUNANA substrate addition by fluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.440nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Hong Kong/68(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50496023(CHEMBL3120197)
Affinity DataIC50: 0.440nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5555/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50496023(CHEMBL3120197)
Affinity DataIC50: 0.450nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5258/2009(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNeuraminidase(Influenza A virus)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 0.450nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Berlin/10/04(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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