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TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623606(CHEMBL5440537)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623607(CHEMBL5440963)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623611(CHEMBL5424952)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623615(CHEMBL5432745)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM297163(US10112941, Example 279 | 2-{8-Fluoro-3-[4-(2H3)me...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of BRD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623605(CHEMBL5401253)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623609(CHEMBL5436475)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623610(CHEMBL5422881)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM439497(US10633379, Example 82 | US10633379, Example 35)
Affinity DataIC50: 0.920nMAssay Description:Inhibition of C-terminal His6-tagged BRD2 BD2 (unknown origin) using H-YSGRGK(Ac)GGK(Ac)GLGK(Ac)-GGAK(Ac)RHRK-Biotin-OH as substrate incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623615(CHEMBL5432745)
Affinity DataIC50: 1nMAssay Description:Inhibition of BRD2 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623602(CHEMBL5422163)
Affinity DataIC50: 1nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707296(US12162878, Compound 56)
Affinity DataIC50: 1.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707295(US12162878, Compound 240)
Affinity DataIC50: 1.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707313(US12162878, Compound 241)
Affinity DataIC50: 1.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707319(US12162878, Compound 251)
Affinity DataIC50: 1.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM296947(US10112941, Example 54 | 2-[3-(Dimethyl-1H-1,2,3-t...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human BRD2 measured by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707307(US12162878, Compound 243)
Affinity DataIC50: 1.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707315(US12162878, Compound 217)
Affinity DataIC50: 1.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707310(US12162878, Compound 250)
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707314(US12162878, Compound 242)
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707315(US12162878, Compound 217)
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707290(US12162878, Compound 213)
Affinity DataIC50: 1.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707294(US12162878, Compound 202)
Affinity DataIC50: 1.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM296886(2-[3-(Dimethyl-1,2-oxazol-4-yl)-5-[oxan-4-yl(pheny...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human BRD2 measured by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707318(US12162878, Compound 212)
Affinity DataIC50: 1.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707312(US12162878, Compound 219)
Affinity DataIC50: 1.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623612(CHEMBL5400310)
Affinity DataIC50: 2nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623613(CHEMBL5439607)
Affinity DataIC50: 2nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707298(US12162878, Compound 184)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707311(US12162878, Compound 41)
Affinity DataIC50: 2.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50576438(CHEMBL4869149)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of recombinant human BRD2 BD2 (348 to 455 residues) expressed in bacterial expression system by bromoscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM192755(TG101209 | US11643396, Example TG101209 | US112797...)
Affinity DataIC50: 2.63nMAssay Description:AlphaScreen is a bead-based, non-radioactive Amplified Luminescent Proximity Homogeneous Assay. The details are not described in this patent.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2023
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707309(US12162878, Compound 193)
Affinity DataIC50: 2.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707297(US12162878, Compound 215)
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50: 3nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50558065(CHEMBL4780530)
Affinity DataIC50: 3nMAssay Description:Inhibition of BRD2 BD1 (unknown origin) using biotinylated JQ1 analog as substrate measured after 20 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50558065(CHEMBL4780530)
Affinity DataIC50: 3nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) using biotinylated JQ1 analog as substrate measured after 20 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623606(CHEMBL5440537)
Affinity DataIC50: 3nMAssay Description:Inhibition of BRD2 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623611(CHEMBL5424952)
Affinity DataIC50: 3nMAssay Description:Inhibition of BRD2 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50092312(Birabresib | MK-8628 | OTX-015)
Affinity DataIC50: 3nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50623604(CHEMBL5403848)
Affinity DataIC50: 3nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM707316(US12162878, Compound 239)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/21/2025
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50459819(CHEMBL4228445)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant N-terminal His6-tagged BRD2 bromodomain 1 (72 to 205 residues) (unknown origin) expressed in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50028142(CHEMBL2177300)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human BRD2 bromodomain 2 by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50520653(CHEMBL4555209)
Affinity DataIC50: 3.5nMAssay Description:Binding affinity to human BRD2 BD1 (72 to 205 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50459819(CHEMBL4228445)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant N-terminal His6-tagged BRD2 bromodomain 2 (349 to 460 residues) (unknown origin) expressed in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of C-terminal His6-tagged BRD2 BD2 (unknown origin) using H-YSGRGK(Ac)GGK(Ac)GLGK(Ac)-GGAK(Ac)RHRK-Biotin-OH as substrate incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM313789(US10167292, Example 33)
Affinity DataIC50: 4nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM543516(US11279703, TABLE 6.37 | US11279703, TABLE 6.199 |...)
Affinity DataIC50: 4.58nMAssay Description:AlphaScreen is a bead-based, non-radioactive Amplified Luminescent Proximity Homogeneous Assay. The details are not described in this patent.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2023
Entry Details
Go to US Patent

TargetBromodomain-containing protein 2(Human)
University of Belgrade

Curated by ChEMBL
LigandPNGBDBM50604624(CHEMBL5206088)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of C-terminal His6-tagged BRD2 BD2 (unknown origin) using H-YSGRGK(Ac)GGK(Ac)GLGK(Ac)-GGAK(Ac)RHRK-Biotin-OH as substrate incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
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