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Report error Found 777 of ic50 data for polymerid = 5516,50006305
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621875(CHEMBL5400397)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621877(CHEMBL5408748)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621883(CHEMBL5431206)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621855(CHEMBL5409024)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621858(CHEMBL5398945)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621880(CHEMBL5428907)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621888(CHEMBL5419830)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621878(CHEMBL5405674)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621884(CHEMBL5399309)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621876(CHEMBL5437496)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621882(CHEMBL5439245)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419721(US10464919, Example 59)
Affinity DataIC50: 0.920nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419799(US10464919, Example 137)
Affinity DataIC50: 0.950nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50204580(N-phenethyl-5-phenyl-6-(4-(2-(pyrrolidin-1-yl)etho...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Ack1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621881(CHEMBL5436567)
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM13216(N-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyeth...)
Affinity DataIC50: 1nMAssay Description:Inhibition of ACK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621879(CHEMBL5434969)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419844(US10464919, Example 182)
Affinity DataIC50: 1.26nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621862(CHEMBL5431312)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419794(US10464919, Example 132)
Affinity DataIC50: 1.31nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419731(US10464919, Example 69)
Affinity DataIC50: 1.32nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419781(US10464919, Example 119)
Affinity DataIC50: 1.38nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419751(US10464919, Example 89)
Affinity DataIC50: 1.48nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419791(US10464919, Example 129)
Affinity DataIC50: 1.65nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419758(US10464919, Example 96)
Affinity DataIC50: 1.75nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419797(US10464919, Example 135)
Affinity DataIC50: 1.75nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419740(US10464919, Example 78)
Affinity DataIC50: 1.87nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621871(CHEMBL5404048)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419832(US10464919, Example 170)
Affinity DataIC50: 1.96nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419755(US10464919, Example 93)
Affinity DataIC50: 1.97nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419761(US10464919, Example 99)
Affinity DataIC50: 1.99nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50246164(N3-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl...)
Affinity DataIC50: 2nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419765(US10464919, Example 103)
Affinity DataIC50: 2.10nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419842(US10464919, Example 180)
Affinity DataIC50: 2.12nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419784(US10464919, Example 122)
Affinity DataIC50: 2.37nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419785(US10464919, Example 123)
Affinity DataIC50: 2.38nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419804(US10464919, Example 142)
Affinity DataIC50: 2.45nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621861(CHEMBL5404162)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419803(US10464919, Example 141)
Affinity DataIC50: 2.62nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of TNK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419796(US10464919, Example 134)
Affinity DataIC50: 2.70nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of ACK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621865(CHEMBL5413451)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419793(US10464919, Example 131)
Affinity DataIC50: 2.81nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419738(US10464919, Example 76)
Affinity DataIC50: 2.86nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621889(CHEMBL5407266)
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419787(US10464919, Example 125)
Affinity DataIC50: 3.18nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM419807(US10464919, Example 145)
Affinity DataIC50: 3.24nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

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