Compile Data Set for Download or QSAR
Report error Found 523 of ic50 data for polymerid = 5445,9915,50002467
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50035236(3-(2-Hydroxycarbamoyl-3-methyl-butyrylamino)-propi...)
Affinity DataIC50: 0.0100nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50035247(2-(2-Hydroxycarbamoyl-3-methyl-butyrylamino)-3-(1H...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50035246(2-(2-Hydroxycarbamoyl-4-methyl-pentanoylamino)-3-(...)
Affinity DataIC50: 0.25nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50251742((S)-2-{(R)-2-[Hydroxy-((2R,3R,4R,5R,6S)-3,4,5-trih...)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50035239(N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-N'-hydroxy...)
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046841(Morpholine-4-carboxylic acid {2-cyclohexyl-1-[1-(2...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50084905({1-[2-Dibenzofuran-3-yl-1-(1H-tetrazol-5-yl)-ethyl...)
Affinity DataIC50: 2.60nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50084905({1-[2-Dibenzofuran-3-yl-1-(1H-tetrazol-5-yl)-ethyl...)
Affinity DataIC50: 2.60nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50035251(2-(2-Hydroxycarbamoyl-3-methyl-butyrylamino)-succi...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50368802(CHEMBL1791097)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407080(CHEMBL2112254)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407074(CHEMBL2112267)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407089(CHEMBL2112253)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50035249(N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-N'-hydroxy...)
Affinity DataIC50: 4.80nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407087(CHEMBL2112258)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407076(CHEMBL2112270)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407075(CHEMBL2112262)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407070(CHEMBL2112268)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046820(4-Methyl-piperazine-1-carboxylic acid {2-cyclohexy...)
Affinity DataIC50: 6nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50084903({[2-Dibenzofuran-3-yl-1-(1H-tetrazol-5-yl)-ethylam...)
Affinity DataIC50: 6nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407071(CHEMBL2112257)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50084897(3-Dibenzofuran-3-yl-2-[3-dibenzofuran-3-yl-2-(phos...)
Affinity DataIC50: 6.40nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50368795(CHEMBL1791129)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50035240((2-Hydroxycarbamoyl-3-methyl-butyrylamino)-acetic ...)
Affinity DataIC50: 6.80nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50159366((2S,4R)-4-Acetylsulfanyl-2-(2,4,5-trifluoro-benzyl...)
Affinity DataIC50: 6.90nMAssay Description:Inhibitory concentration against human ECE-1 by RIAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50368810(CHEMBL1791125)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407072(CHEMBL2112269)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50105264(2-(2-Benzyl-3-hydroxycarbamoyl-propionylamino)-pro...)
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM21641(2-(2-benzyl-3-sulfanylpropanamido)acetic acid | CH...)
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50064110(CHEMBL147847 | 2-{2-[(S)-5-(2,4-Difluoro-phenyl)-2...)
Affinity DataIC50: 8nMAssay Description:In Vitro inhibition of recombinant human endothelin converting enzyme-1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50119751(2-{[1-(2-Mercapto-4-methyl-pentanoylamino)-cyclope...)
Affinity DataIC50: 9.5nMAssay Description:In vitro inhibition of Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50119742(2-{[1-(2-Mercapto-4-methyl-pentanoylamino)-cyclope...)
Affinity DataIC50: 9.80nMAssay Description:In vitro inhibition of Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50119742(2-{[1-(2-Mercapto-4-methyl-pentanoylamino)-cyclope...)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of Homo sapiens (human) endothelin converting enzyme-1More data for this Ligand-Target Pair
In DepthDetails Article

TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50171626(CHEMBL381643 | ECE Inhibitor, 11 | 5-(3,3-Dimethyl...)
Affinity DataIC50: 10nMAssay Description:Inhibition assay using ECE.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM97371(ECE Inhibitor, 14)
Affinity DataIC50: 10nMAssay Description:Inhibition assay using ECE.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50159365((3R,5S)-5-{[(2,5-difluorobenzyl)amino]methyl}-1-(5...)
Affinity DataIC50: 10.4nMAssay Description:Inhibitory concentration against human ECE-1 by RIAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50035235(N-[1-(Carbamoylmethyl-carbamoyl)-ethyl]-N''-hydrox...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against human bronchiolar smooth muscle Endothelin-converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50091878((S)-3-Biphenyl-4-yl-2-{[1-((S)-2-mercapto-3-methox...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of human Endothelin converting Enzyme-1 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50091882(3-Biphenyl-4-yl-2-{[1-(2-mercapto-pentanoylamino)-...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of human Endothelin converting Enzyme-1 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50091882(3-Biphenyl-4-yl-2-{[1-(2-mercapto-pentanoylamino)-...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibitory activity was tested against Endothelin converting enzyme 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50091882(3-Biphenyl-4-yl-2-{[1-(2-mercapto-pentanoylamino)-...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50368798(CHEMBL1791120)
Affinity DataIC50: 11nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50368814(CHEMBL1791126)
Affinity DataIC50: 11nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407088(CHEMBL2112255)
Affinity DataIC50: 11nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50488971(CHEMBL2297562)
Affinity DataIC50: 11nMAssay Description:Inhibition of Homo sapiens (human) endothelin converting enzyme-1More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article

TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50488983(CHEMBL2297552)
Affinity DataIC50: 11nMAssay Description:Inhibition of Homo sapiens (human) endothelin converting enzyme-1More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article

TargetEndothelin-converting enzyme 1(Human)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50098118((2S,4R)-4-Mercapto-2-(2,4,5-trifluoro-benzyloxymet...)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against human ECE-1 by RIAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50407086(CHEMBL2112265)
Affinity DataIC50: 12nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046842(3-{4-[2-(2-tert-Butoxycarbonylamino-3-methyl-penta...)
Affinity DataIC50: 13nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin-converting enzyme 1(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046857([1-(1-{1-[1-Hydroxy-2-(4-hydroxy-butylcarbamoyl)-e...)
Affinity DataIC50: 13nMAssay Description:Inhibition of conversion of big endothelial-1 (Big ET-1) to ET-1 by endothelin converting enzyme(ECE) in rat lung membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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