Compile Data Set for Download or QSAR
Report error Found 94 of ic50 data for polymerid = 5373
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50033762(Gallinamide A)
Affinity DataIC50: 22nMAssay Description:Inhibition of Plasmodium falciparum D10 trophozite lysates FP-3 pretreated with compound for 1 hr followed by labeling with Cy5-DCG04 for 1 hr by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50448248(CHEMBL3120847)
Affinity DataIC50: 60nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513155(CHEMBL4434685)
Affinity DataIC50: 79nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50286441(Ac-LLR-CHO | Ac-Leu-Leu-Arg-H | (S)-2-((S)-2-Acety...)
Affinity DataIC50: 87nMAssay Description:Inhibition of Cysteine protease falcipain-3 in Plasmodium falciparum HB3 infected erythrocytes by Z-Phe-Arg-AMC substrate hydrolysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50286441(Ac-LLR-CHO | Ac-Leu-Leu-Arg-H | (S)-2-((S)-2-Acety...)
Affinity DataIC50: 98nMAssay Description:Inhibition of Cysteine protease falcipain-3 in Plasmodium falciparum HB3-leuR1 mutant infected erythrocytes by Z-Phe-Arg-AMC substrate hydrolysis ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513158(CHEMBL4439637)
Affinity DataIC50: 112nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50: 116nMAssay Description:Inhibition of Plasmodium falciparum FP3 using Z-Leu-Arg-AMC as substrate incubated for 30 mins by spectrofluorometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513162(CHEMBL4467013)
Affinity DataIC50: 117nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50461247(CHEMBL4228861)
Affinity DataIC50: 117nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513161(CHEMBL4472824)
Affinity DataIC50: 131nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM12042(L-trans-3-Carboxyoxiran-2-carbonyl-L-leucylagmatin...)
Affinity DataIC50: 136nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513163(CHEMBL4442854)
Affinity DataIC50: 228nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513168(CHEMBL4437416)
Affinity DataIC50: 407nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513165(CHEMBL4475837)
Affinity DataIC50: 459nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513166(CHEMBL4527228)
Affinity DataIC50: 480nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50: 482nMAssay Description:Inhibition of Plasmodium falciparum falcipain 3 incubated with compound for 10 mins before addition of 25 uM Z-Leu-Arg-AMC substrate by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513156(CHEMBL4442674)
Affinity DataIC50: 484nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513159(CHEMBL4516951)
Affinity DataIC50: 490nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50448247(CHEMBL3120848)
Affinity DataIC50: 520nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50448261(CHEMBL3120834)
Affinity DataIC50: 540nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513157(CHEMBL4555968)
Affinity DataIC50: 547nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513167(CHEMBL4564002)
Affinity DataIC50: 851nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50448260(CHEMBL3120835)
Affinity DataIC50: 910nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50513160(CHEMBL4456644)
Affinity DataIC50: 2.57E+3nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His-tagged falcipain-3 (33 residues) expressed in Escherichia coli M15 pREP4 using Z-Leu-Arg-AMC as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50448246(CHEMBL3120849)
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50621181(CHEMBL5434874)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of Plasmodium falciparum FP3 using Z-Leu-Arg-AMC as substrate incubated for 30 mins by spectrofluorometry analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529719(CHEMBL1302947)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529721(CHEMBL4444541)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529712(CHEMBL4451728)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529721(CHEMBL4444541)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529717(CHEMBL4578038)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529719(CHEMBL1302947)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529712(CHEMBL4451728)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529722(CHEMBL4582464)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529714(CHEMBL4458321)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529720(CHEMBL4551614)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529713(CHEMBL4449400)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529714(CHEMBL4458321)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529715(CHEMBL4471644)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529716(CHEMBL1584095)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529717(CHEMBL4578038)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529718(CHEMBL4582597)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529713(CHEMBL4449400)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529715(CHEMBL4471644)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529716(CHEMBL1584095)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529718(CHEMBL4582597)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529720(CHEMBL4551614)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50529722(CHEMBL4582464)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50621179(CHEMBL5398485)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of Plasmodium falciparum FP3 using Z-Leu-Arg-AMC as substrate incubated for 30 mins by spectrofluorometry analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University of Petroleum and Energy Studies

Curated by ChEMBL
LigandPNGBDBM50621182(CHEMBL5400091)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of Plasmodium falciparum FP3 using Z-Leu-Arg-AMC as substrate incubated for 30 mins by spectrofluorometry analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
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