Compile Data Set for Download or QSAR
Report error Found 538 of ic50 data for polymerid = 5163,5165,50001134,50005686
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50147093(6-[(Z)-AMINO(IMINO)METHYL]-N-[4-(AMINOMETHYL)PHENY...)
Affinity DataIC50: 0.620nMAssay Description:Inhibition of uPA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194745(diphenyl 1-[(N-2-thiophenesulfonyl-D-seryl)-L-alan...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194741(diphenyl 1-[(N-benzenesulfonyl-D-seryl)-L-alanyl]a...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088982(CHEMBL160253 | CHEMBL367004 | N-[1-(1-Carbamimidoy...)
Affinity DataIC50: 3.10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228418(methyl 1-(diphenoxyphosphoryl)-2-(4-guanidinopheny...)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228412(methyl 1-(bis(4-acetamidophenoxy)phosphoryl)-2-(4g...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194743(diphenyl 1-[(N-alpha-toluenesulfonyl-D-seryl)-L-al...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228425(di-(4-acetamidophenyl) 1-(methylsulfonylamino)-2-(...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194743(diphenyl 1-[(N-alpha-toluenesulfonyl-D-seryl)-L-al...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
University of Michigan

LigandPNGBDBM92479(Tannic Acid, A | Tannic acid)
Affinity DataIC50: 4.10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228420(di-(4-acetamidophenyl) 1-(benzyloxycarbonylamino)-...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50145689([1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194737(diphenyl 1-[(N-o-methylbenzoyl-D-seryl)-L-alanyl]a...)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194746(diphenyl 1-[(N-o-methylbenzoyl-D-seryl)-L-alanyl]a...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194742(diphenyl 1-[(N-benzyl-D-seryl)-L-alanyl]amino-2-(4...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088978(N-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcarb...)
Affinity DataIC50: 5.10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194734(diphenyl 1-[(N-p-methoxybenzenesulfonyl-D-seryl)-L...)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194744(diphenyl 1-[(N-naphthalenesulfonyl-D-seryl)-L-alan...)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194736(diphenyl 1-[(N-o,o-dimethylbenzoyl-D-seryl)-L-alan...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194735(diphenyl 1-[(N-p-cyanobenzenesulfonyl-D-seryl)-L-a...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM92479(Tannic Acid, A | Tannic acid)
Affinity DataIC50: 6.60nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194738(diphenyl 1-[(N-p-bromobenzenesulfonyl-D-seryl)-L-a...)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228421(diphenyl 1-(methylsulfonylamino)-2-(4-guanidinophe...)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194732(di-(4-acetamidophenyl) 1-[(N-benzyloxycarbonyl-D-s...)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194739(diphenyl 1-[(N-2-thienyl-D-seryl)-L-alanyl]amino-2...)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194740(diphenyl 1-[(N-p-methylbenzoyl-D-seryl)-L-alanyl]a...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228410(diphenyl 1-(benzyloxycarbonylamino)-2-(4-guanidino...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228414(diphenyl 1-acetamido-2-(4-guanidinophenyl)ethylpho...)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228417(diphenyl 1-(o-toluenesulfonylamino)-2-(4-guanidino...)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194733(diphenyl 1-[(N-1-adamantanyl-D-seryl)-L-alanyl])am...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
University of Michigan

LigandPNGBDBM50228412(methyl 1-(bis(4-acetamidophenoxy)phosphoryl)-2-(4g...)
Affinity DataIC50: 8nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228423(ethyl 1-(diphenoxyphosphoryl)-2-(4-guanidinophenyl...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM92485(CDE-066 | US9120744, CDE-066)
Affinity DataIC50: 10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
University of Michigan

LigandPNGBDBM92485(CDE-066 | US9120744, CDE-066)
Affinity DataIC50: 10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088984(2-Benzenesulfonylamino-N-[1-(1-carbamimidoyl-2-hyd...)
Affinity DataIC50: 10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
University of Michigan

LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50: 10nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured immediatelyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088979({(R)-2-[2-((S)-1-Carbamimidoyl-2-hydroxy-piperidin...)
Affinity DataIC50: 11nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
University of Michigan

LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50: 11nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 8 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088985({2-[2-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 12nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
University of Michigan

LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50: 12nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM92486(CDE-082 | US9120744, CDE-082)
Affinity DataIC50: 14nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50301972(2-(6-(5-amino-3'-(aminomethyl)biphenyl-3-yloxy)-4-...)
Affinity DataIC50: 15nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50542728(CHEMBL4635912)
Affinity DataIC50: 16nMAssay Description:Inhibition of human urokinase using fluorescent peptide as substrate by florescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088977({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 19nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Rat)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228418(methyl 1-(diphenoxyphosphoryl)-2-(4-guanidinopheny...)
Affinity DataIC50: 19.5nMAssay Description:Inhibition of rat uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM92487(CDE-031 | US9120744, CDE-031)
Affinity DataIC50: 20nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50231520(CHEMBL252937 | US8476306, 6.12 | (R)-N-[(S)-1-(4-c...)
Affinity DataIC50: 20nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50542731(CHEMBL4642845)
Affinity DataIC50: 20nMAssay Description:Inhibition of human uPA using fluorescent peptide as substrate by florescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50542732(CHEMBL4647925)
Affinity DataIC50: 20nMAssay Description:Inhibition of human uPA using fluorescent peptide as substrate by florescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088987({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 23nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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