Compile Data Set for Download or QSAR
Report error Found 8 of ic50 data for polymerid = 50007839
TargetToll-like receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50552135(CHEMBL4303210)
Affinity DataIC50: 54nMAssay Description:Inhibition of Rho-Pam3 binding to TLR1 (unknown origin)/human TLR2 expressed in HEK293 cells incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetToll-like receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50552138(CHEMBL3935646)
Affinity DataIC50: 580nMAssay Description:Antagonist activity at TLR1/TLR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetToll-like receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM34883(ethyl 5-[2-oxidanylidene-2-[2,3,4-tris(oxidanyl)ph...)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human TLR1/TLR2More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetToll-like receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50543142(CHEMBL4641633)
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonist activity at TLR1 in human PBMC assessed as inhibition of Pam3CSK4-induced TNFalpha production preincubated for 30 mins followed by Pam3CSK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetToll-like receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50552138(CHEMBL3935646)
Affinity DataIC50: 9.10E+3nMAssay Description:Antagonist activity at human TLR1/TLR2More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetToll-like receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50622099(CHEMBL4227186)
Affinity DataIC50: 1.97E+4nMAssay Description:Antagonist activity at TLR1/TLR2 in HEK-Blue hTLR2 cellsMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetToll-like receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM111024(US8614253, 3-63 | US8614253, 3-55 | US9241942, 3-6...)
Affinity DataIC50: 2.42E+4nMAssay Description:Antagonist activity at TLR1/TLR2 in HEK-Blue hTLR2 cellsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetToll-like receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50463543(CHEMBL4249593)
Affinity DataIC50: 4.58E+4nMAssay Description:Antagonist activity at FLAG-tagged human TLR2/TLR1 expressed in HEK293 cells co-expressing pGL3-Elam.luc assessed as inhibition of Pam3CSK4-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed