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Report error Found 66 of ic50 data for polymerid = 50007369
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50568523(CHEMBL4875015)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of N-terminal His-SUMO tagged human LSD1 (172 to 852 residues)/His-tagged CoREST (286 to 482 residues) expressed in Escherichia coli BL21 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50153586(CHEMBL3775474 | US10053456, 120 | US9718814, 71 | ...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50410785(CHEMBL5291155)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50410784(CHEMBL5280566)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50410789(CHEMBL5277056)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50621408(CHEMBL5399284)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50410788(CHEMBL5281376)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50621404(CHEMBL5421067)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50403543(CHEMBL5276713)
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human LSD1/CoREST by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50410786(CHEMBL5270114)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498143(CHEMBL3407602)
Affinity DataIC50: 31nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498128(CHEMBL3410944)
Affinity DataIC50: 35nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498142(CHEMBL3407601)
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM256729(US9487511, 125 | US10053456, 125 | US9718814, 125 ...)
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498137(CHEMBL3410941)
Affinity DataIC50: 47nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50410787(CHEMBL5270703)
Affinity DataIC50: 64nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498150(CHEMBL3407599)
Affinity DataIC50: 79nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50621401(CHEMBL5403890)
Affinity DataIC50: 82nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50568517(CHEMBL4848459)
Affinity DataIC50: 90nMAssay Description:Inhibition of human LSD1/CoREST expressed in Escherichia coli using monomethylated H3-K4 peptide as substrate preincubated for 15 mins followed by su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498135(CHEMBL3407603)
Affinity DataIC50: 94nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498134(CHEMBL3407605)
Affinity DataIC50: 96nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50621404(CHEMBL5421067)
Affinity DataIC50: 98nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498147(CHEMBL3407604)
Affinity DataIC50: 101nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50458056(CHEMBL4208031)
Affinity DataIC50: 107nMAssay Description:Inhibition of recombinant human LSD1/CoREST preincubated for 5 mins followed by ART-(N,N-dimethyl-K)-QTARKSTGGKAPRKQLA substrate addition measured af...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50458056(CHEMBL4208031)
Affinity DataIC50: 107nMAssay Description:Inhibition of recombinant human LSD1/CoREST preincubated for 5 mins followed by ART-(N,N-dimethyl-K)-QTARKSTGGKAPRKQLA substrate addition measured af...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498141(CHEMBL3407597)
Affinity DataIC50: 118nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498130(CHEMBL3407600)
Affinity DataIC50: 121nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498140(CHEMBL3407596)
Affinity DataIC50: 123nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50458055(CHEMBL4214605)
Affinity DataIC50: 136nMAssay Description:Inhibition of recombinant human LSD1/CoREST preincubated for 5 mins followed by ART-(N,N-dimethyl-K)-QTARKSTGGKAPRKQLA substrate addition measured af...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50458055(CHEMBL4214605)
Affinity DataIC50: 136nMAssay Description:Inhibition of recombinant human LSD1/CoREST preincubated for 5 mins followed by ART-(N,N-dimethyl-K)-QTARKSTGGKAPRKQLA substrate addition measured af...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498144(CHEMBL3407608)
Affinity DataIC50: 158nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50621403(CHEMBL5433869)
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498133(CHEMBL3407606)
Affinity DataIC50: 173nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498151(CHEMBL3407598)
Affinity DataIC50: 178nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498132(CHEMBL3407612)
Affinity DataIC50: 187nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50621405(CHEMBL5418529)
Affinity DataIC50: 230nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498131(CHEMBL3407613)
Affinity DataIC50: 230nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498149(CHEMBL3407594)
Affinity DataIC50: 248nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498127(CHEMBL3407607)
Affinity DataIC50: 251nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498145(CHEMBL3407593)
Affinity DataIC50: 258nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498152(CHEMBL3407611)
Affinity DataIC50: 263nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50153587(US9487511, 82 | CHEMBL3775248 | US10053456, 82 | U...)
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50621406(CHEMBL5436851)
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498129(CHEMBL3407609)
Affinity DataIC50: 279nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50568518(CHEMBL4877195)
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human KDM1A/CoREST expressed in Escherichia coli using mono-methylated H3-K4 peptide as substrate preincubated for 15 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50548040(CHEMBL4791172)
Affinity DataIC50: 330nMAssay Description:Inhibition of LSD1/FLAG-tagged CoREST (unknown origin) expressed in HEK293F cells using diMeK4H3(1 to 21 residues) as substrate preincubated for 5 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50610592(CHEMBL5272967)
Affinity DataIC50: 330nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 expressed in Escherichia coli using ARTK (Me)-2QTARKSTGGKAPRKQLA as substrate/FLAG-tagged CoREST trans...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498139(CHEMBL3407592)
Affinity DataIC50: 350nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498138(CHEMBL3410945)
Affinity DataIC50: 352nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetREST corepressor 1(Human)
Key Laboratory of Henan Provinc

Curated by ChEMBL
LigandPNGBDBM50498136(CHEMBL3410942)
Affinity DataIC50: 554nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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