Compile Data Set for Download or QSAR
Report error Found 6 of ic50 data for polymerid = 50006913
TargetBromodomain-containing protein 8(Human)
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50510872(CHEMBL4303404)
Affinity DataIC50: 1.50E+4nMAssay Description:Displacement of biotinylated JQ1 from BRD8 bromodomain (unknown origin) incubated for 20 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 8(Human)
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50510872(CHEMBL4303404)
Affinity DataIC50: 1.50E+4nMAssay Description:Binding affinity to BRD8 bromodomain (unknown origin) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 8(Human)
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200385(CHEMBL3959584)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged BRD8 bromodomain-1 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 8(Human)
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200384(CHEMBL3968533 | US9763922, Example 299)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged BRD8 bromodomain-1 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 8(Human)
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50269847(CHEMBL4097025)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of biotinylated histone H3K14 peptide ligand from recombinant His-tagged BRD8 bromodomain-1 (unknown origin) measured after 10 mins by T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 8(Human)
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50269849(CHEMBL4076748)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of biotinylated histone H3K14 peptide ligand from recombinant His-tagged BRD8 bromodomain-1 (unknown origin) measured after 10 mins by T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed