Compile Data Set for Download or QSAR
Report error Found 75 of ic50 data for polymerid = 50006411
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544215(CHEMBL4637689)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544211(CHEMBL4641682)
Affinity DataIC50: 0.0870nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544227(CHEMBL4634501)
Affinity DataIC50: 0.170nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50286578(CHEMBL4170617)
Affinity DataIC50: 0.670nMAssay Description:Inhibition of human recombinant HDAC3/GST-tagged NCOR1 DAD (397 to 503 residues) expressed in baculovirus expression system after 30 mins by fluoresc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544217(CHEMBL4644307)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544213(CHEMBL4647458)
Affinity DataIC50: 2nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544212(CHEMBL4632775)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544223(CHEMBL4637836)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50286560(CHEMBL4163681)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human recombinant HDAC3/GST-tagged NCOR1 DAD (397 to 503 residues) expressed in baculovirus expression system after 30 mins by fluoresc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of human recombinant HDAC3/GST-tagged NCOR1 DAD (397 to 503 residues) expressed in baculovirus expression system after 30 mins by fluoresc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437809(CHEMBL2407717)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437812(CHEMBL2407723)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544226(CHEMBL4632449)
Affinity DataIC50: 13nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437821(CHEMBL2407736)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544225(CHEMBL4641904)
Affinity DataIC50: 15nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437816(CHEMBL2407719)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50361170(CHEMBL4159366)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant HDAC3/GST-tagged NCOR1 (397 to 503 residues) co-expressed in insect cells using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544224(CHEMBL4644721)
Affinity DataIC50: 20nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544228(CHEMBL4647164)
Affinity DataIC50: 23nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437813(CHEMBL2407722)
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437822(CHEMBL2407735)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437827(CHEMBL2407730)
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437814(CHEMBL2407721)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437826(CHEMBL2407731)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50361177(CHEMBL4160840)
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant HDAC3/GST-tagged NCOR1 (397 to 503 residues) co-expressed in insect cells using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544214(CHEMBL4633968)
Affinity DataIC50: 50nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 51nMAssay Description:Inhibition of human recombinant HDAC3/GST tagged NCOR1 (397 to 503 residues) expressed in insect cells using Ac-Leu-Gly-Lys(Ac)-AMC as substrate prei...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437815(CHEMBL2407720)
Affinity DataIC50: 52nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 54nMAssay Description:Inhibition of recombinant human GST-fused HDAC3/NCOR1 (397 to 503 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Ac)-A...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437818(CHEMBL2407716)
Affinity DataIC50: 63nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437825(CHEMBL2407732)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50565547(CHEMBL4781177)
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant human GST-fused HDAC3/NCOR1 (397 to 503 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Ac)-A...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437817(CHEMBL2407718)
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437823(CHEMBL2407734)
Affinity DataIC50: 83nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544221(CHEMBL4639586)
Affinity DataIC50: 90nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437824(CHEMBL2407733)
Affinity DataIC50: 104nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50565548(CHEMBL4790998)
Affinity DataIC50: 106nMAssay Description:Inhibition of recombinant human GST-fused HDAC3/NCOR1 (397 to 503 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Ac)-A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50437833(CHEMBL2407742)
Affinity DataIC50: 111nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544222(CHEMBL4646763)
Affinity DataIC50: 120nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50525180(CHEMBL4446236)
Affinity DataIC50: 136nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544218(CHEMBL4636534)
Affinity DataIC50: 150nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50525179(CHEMBL4450474)
Affinity DataIC50: 215nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50544219(CHEMBL4644575)
Affinity DataIC50: 230nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50242817(CHEMBL4087968 | US20240150300, Compound Chidamide)
Affinity DataIC50: 234nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50361171(CHEMBL4175555)
Affinity DataIC50: 234nMAssay Description:Inhibition of human recombinant HDAC3/GST-tagged NCOR1 (397 to 503 residues) co-expressed in insect cells using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50121210(CHEMBL3622374)
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human HDAC3/GST-tagged NCOR1 DAD (397 to 503 residues) expressed in baculovirus expression system using Fluor de Lys as sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50121210(CHEMBL3622374)
Affinity DataIC50: 240nMAssay Description:Inhibition of human recombinant HDAC3/GST-tagged NCOR1 DAD (397 to 503 residues) expressed in baculovirus expression system by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50121211(CHEMBL3622375)
Affinity DataIC50: 260nMAssay Description:Inhibition of human recombinant HDAC3/GST-tagged NCOR1 DAD (397 to 503 residues) expressed in baculovirus expression system by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50121211(CHEMBL3622375)
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant human HDAC3/GST-tagged NCOR1 DAD (397 to 503 residues) expressed in baculovirus expression system using Fluor de Lys as sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor corepressor 1(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50525178(CHEMBL4437852)
Affinity DataIC50: 274nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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