Report error Found 57 of ic50 data for polymerid = 50004562,50007540
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 14.4nMAssay Description:Inhibition of human STK39 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 17.2nMAssay Description:Inhibition of human STK39 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of STLK3 (unknown origin)More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of STLK3 (unknown origin)More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human STK39 using MBP substrateMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 2.11E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 2.82E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 3.56E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 3.69E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical and Dental University (Tmdu)
Curated by ChEMBL
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
