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TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human TSSK2 using KKKVSRSGLYRSPSMPENLNRPR as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human TSSK2 using KKKVSRSGLYRSPSMPENLNRPR as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50: 30.6nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50335188(CHEMBL1650551 | CHEMBL1650545 | N-[3-[(3,3-Difluor...)
Affinity DataIC50: 100nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50335188(CHEMBL1650551 | CHEMBL1650545 | N-[3-[(3,3-Difluor...)
Affinity DataIC50: 100nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50329198(CHEMBL1650533 | 2-{ethyl[(5-{[6-methyl-3-(1H-pyraz...)
Affinity DataIC50: 100nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50460773(CHEMBL4227082)
Affinity DataIC50: 500nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50460767(CHEMBL4228240)
Affinity DataIC50: 500nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50582077(CHEMBL5085753)
Affinity DataIC50: 944nMAssay Description:Inhibition of TSSK2 (unknown origin) by Z-lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50462709(CHEMBL4245507)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50433476(CHEMBL2381116)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50348621(CHEMBL1270795)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50499634(CHEMBL3741589)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TSSK2 using [KKKVSRSGLYRSPSMPENLNRPR] as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50519662(CHEMBL4438748)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant full-length human TSSK2 using KKKVSRSGLYRSP as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50433761(CHEMBL2381601)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50434485(CHEMBL2385543)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50362169(CHEMBL1938680)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50359359(CHEMBL1929238)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50030881(CHEMBL3356117)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant full length human His-tagged STK22B expressed in baculovirus expression system using serine/threonine-04 peptide as substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed