Compile Data Set for Download or QSAR
Report error Found 13 of ic50 data for polymerid = 50003979
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311193(US10155760, Example 37 | (S)-1-(2-(difluoromethyl)...)
Affinity DataIC50: 56nMAssay Description:Inhibition of CRIK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311212(US10155760, Example 68 | (S)-methyl (5-((2-amino-2...)
Affinity DataIC50: 60nMAssay Description:Inhibition of CRIK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311210(US10155760, Example 66 | (S)-methyl (5-((2-amino-2...)
Affinity DataIC50: 90nMAssay Description:Inhibition of CRIK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50573682(CHEMBL4872886)
Affinity DataIC50: 120nMAssay Description:Inhibition of CRIK (unknown origin) by Kinomescan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311267(US10155760, Example 123 | (S)-1-((2′,6-bis(d...)
Affinity DataIC50: 410nMAssay Description:Inhibition of CRIK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 458nMAssay Description:Inhibition of human STK21 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311266(US10155760, Example 122 | (S)-1-((4-(difluoromethy...)
Affinity DataIC50: 750nMAssay Description:Inhibition of CRIK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50045333(CHEBI:90705 | SB-203580)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human CITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human STK21 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311268(US10155760, Example 124 | (S)-1-((2′,4-bis(d...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of CRIK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311381(US10155760, Example 238 | (S)-1-((4-chloro-2′...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CRIK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50462710(CHEMBL4251324)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of CIT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCitron Rho-interacting kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50462709(CHEMBL4245507)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CIT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed